Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50040301
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194496BDBM194496(BDBM50392261 | US9200020, Table 3 compound 5)
Affinity DataKi:  70nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194501BDBM194501(BDBM50392263 | US9200020, Table 3 compound 10)
Affinity DataKi:  70nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194492BDBM194492(US9200020, Table 3 compound 1 | BDBM50392258)
Affinity DataKi:  100nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194494BDBM194494(BDBM50392260 | US9200020, Table 3 compound 3)
Affinity DataKi:  100nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194500BDBM194500(BDBM50392266 | US9200020, Table 3 compound 9)
Affinity DataKi:  100nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194499BDBM194499(BDBM50392265 | US9200020, Table 3 compound 8)
Affinity DataKi:  150nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194502BDBM194502(US9200020, Table 3 compound 11 | BDBM50392267)
Affinity DataKi:  200nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194493BDBM194493(US9200020, Table 3 compound 2 | BDBM50392259)
Affinity DataKi:  500nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194497BDBM194497(BDBM50392262 | US9200020, Table 3 compound 6)
Affinity DataKi:  600nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194498BDBM194498(BDBM50392264 | US9200020, Table 3 compound 7)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60890BDBM60890(BDBM50392251 | US9200020, Table 3 compound 5B)
Affinity DataKi:  2.40E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60886BDBM60886(US9200020, Table 3, Compound 1B | BDBM50392247)
Affinity DataKi:  2.60E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60897BDBM60897(US9200020, Table 3 compound 11B | BDBM50392257)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194491BDBM194491(US9200020, Table 1, Compound 2 | BDBM50392245)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60894BDBM60894(BDBM50392256 | US9200020, Table 3 compound 9B)
Affinity DataKi:  5.40E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60896BDBM60896(BDBM50392253 | US9200020, Table 3 compound 10B)
Affinity DataKi:  5.50E+3nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60888BDBM60888(US9200020, Table 3, Compound 3B | BDBM50392249)
Affinity DataKi:  2.20E+4nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60891BDBM60891(BDBM50392252 | US9200020, Table 3 compound 6B)
Affinity DataKi:  2.90E+4nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60892BDBM60892(BDBM50392254 | US9200020, Table 3 compound 7B)
Affinity DataKi:  3.20E+4nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 194495BDBM194495(BDBM50392250 | US9200020, Table 3 compound 4)
Affinity DataKi:  3.50E+4nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392246BDBM50392246(CHEMBL2153499)
Affinity DataKi:  4.00E+4nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 60887BDBM60887(US9200020, Table 3, Compound 2B | BDBM50392248)
Affinity DataKi: >2.00E+5nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Human)
Academy of Sciences of The Czech Republic

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50392255BDBM50392255(CHEMBL2153493)
Affinity DataKi: >2.40E+5nMAssay Description:Inhibition of human HGPRT using Prib-PP as substrate by spectrophotometric assay in presence of guanineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed