Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50040125
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070942BDBM50070942((-)-Epigallocatechin-3-o-gallate | (-)-Epigallocat...)
Affinity DataKi:  28nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389497BDBM50389497(CHEMBL1564869)
Affinity DataKi:  230nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389487BDBM50389487(CHEMBL2063048)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389487BDBM50389487(CHEMBL2063048)
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of Spiroplasma sp. MQ1 SssI methyltransferase-mediated DNA cytosine methylation using pUC18 as substrate and [3H]CH3-SAM measured up to 10...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389488BDBM50389488(CHEMBL2063060)
Affinity DataKi:  3.60E+3nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389495BDBM50389495(CHEMBL2063052)
Affinity DataKi:  1.00E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389498BDBM50389498(CHEMBL2063050)
Affinity DataKi:  1.50E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389489BDBM50389489(CHEMBL2063059)
Affinity DataKi:  2.00E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetDNA (cytosine-5)-methyltransferase 1(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389487BDBM50389487(CHEMBL2063048)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of DNMT1 in human HeLa cell nuclear extract assessed as methylated substrate level by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389481BDBM50389481(CHEMBL2063056)
Affinity DataKi:  2.30E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389494BDBM50389494(CHEMBL2063053)
Affinity DataKi:  2.60E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389491BDBM50389491(CHEMBL2063057)
Affinity DataKi:  3.30E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389490BDBM50389490(CHEMBL2063058)
Affinity DataKi:  3.50E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389503BDBM50389503(CHEMBL2063044)
Affinity DataKi:  5.00E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389482BDBM50389482(CHEMBL1699292)
Affinity DataKi:  7.00E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389501BDBM50389501(CHEMBL2063046)
Affinity DataKi:  8.30E+4nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389502BDBM50389502(CHEMBL2063045)
Affinity DataKi:  1.12E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389492BDBM50389492(CHEMBL2063055)
Affinity DataKi:  1.35E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389505BDBM50389505(CHEMBL2063041)
Affinity DataKi:  1.70E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389499BDBM50389499(CHEMBL2063049)
Affinity DataKi:  2.50E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389493BDBM50389493(CHEMBL2063054)
Affinity DataKi:  4.00E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389504BDBM50389504(CHEMBL2063043)
Affinity DataKi:  4.40E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389496BDBM50389496(CHEMBL472604)
Affinity DataKi:  5.50E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389509BDBM50389509(CHEMBL2063042)
Affinity DataKi:  7.00E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389506BDBM50389506(CHEMBL2063064)
Affinity DataKi:  8.00E+5nMAssay Description:Uncompetitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Cornish-Bowden's plot analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389500BDBM50389500(CHEMBL2063047)
Affinity DataKi:  9.60E+5nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389485BDBM50389485(CHEMBL2063066)
Affinity DataKi:  1.00E+6nMAssay Description:Uncompetitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Cornish-Bowden's plot analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389483BDBM50389483(CHEMBL2063063)
Affinity DataKi:  3.40E+6nMAssay Description:Uncompetitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Cornish-Bowden's plot analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389508BDBM50389508(CHEMBL1230389)
Affinity DataKi:  5.50E+6nMAssay Description:Competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389486BDBM50389486(CHEMBL2063062)
Affinity DataKi:  5.60E+6nMAssay Description:Uncompetitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Cornish-Bowden's plot analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389484BDBM50389484(CHEMBL2063065)
Affinity DataKi:  6.00E+6nMAssay Description:Uncompetitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Cornish-Bowden's plot analysi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetOrphan methyltransferase M.SssI(Spiroplasma monobiae strain MQ-1)
Polish Academy of Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50389507BDBM50389507(CHEMBL2063051)
Affinity DataKi:  6.40E+6nMAssay Description:Non-competitive inhibition of Spiroplasma sp. MQ1 SssI methyltransferase using pUC18 as substrate measured for 10 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed