Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50040536
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395751(CHEMBL2164507)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395751(CHEMBL2164507)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395753(CHEMBL2164499)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395753(CHEMBL2164499)
Affinity DataKi:  8nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395743(CHEMBL2164832)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395765(CHEMBL2164503)
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395752(CHEMBL2164500)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395744(CHEMBL2164831)
Affinity DataKi:  44nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395749(CHEMBL2164826)
Affinity DataIC50: 47nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395763(CHEMBL2164505)
Affinity DataIC50: 47nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395767(CHEMBL2164501)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395744(CHEMBL2164831)
Affinity DataIC50: 72nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395764(CHEMBL2164504)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395758(CHEMBL2164823)
Affinity DataIC50: 110nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395745(CHEMBL2164830)
Affinity DataIC50: 111nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395752(CHEMBL2164500)
Affinity DataKi:  121nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395750(CHEMBL2164508)
Affinity DataIC50: 129nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395748(CHEMBL2164827)
Affinity DataIC50: 140nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395758(CHEMBL2164823)
Affinity DataKi:  202nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395755(CHEMBL2164494)
Affinity DataIC50: 213nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395754(CHEMBL2164497)
Affinity DataIC50: 220nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395766(CHEMBL2164502)
Affinity DataIC50: 239nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395749(CHEMBL2164826)
Affinity DataKi:  249nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395774(CHEMBL2164834)
Affinity DataIC50: 251nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395746(CHEMBL2164829)
Affinity DataIC50: 273nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395750(CHEMBL2164508)
Affinity DataKi:  286nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395755(CHEMBL2164494)
Affinity DataKi:  392nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395773(CHEMBL2164835)
Affinity DataIC50: 525nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395742(CHEMBL2164833)
Affinity DataIC50: 700nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395754(CHEMBL2164497)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]-ghrelin from human GHSR1 expressed in CHO-CREluc cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395771(CHEMBL2164493)
Affinity DataIC50: 1.16E+3nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395770(CHEMBL2164495)
Affinity DataIC50: 1.18E+3nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395747(CHEMBL2164828)
Affinity DataIC50: 1.39E+3nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395772(CHEMBL2164492)
Affinity DataIC50: 1.47E+3nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395756(CHEMBL2164825)
Affinity DataIC50: 2.54E+3nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395762(CHEMBL2164506)
Affinity DataIC50: 2.78E+3nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395749(CHEMBL2164826)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395757(CHEMBL2164824)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395768(CHEMBL2164498)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395759(CHEMBL2164822)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395769(CHEMBL2164496)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395761(CHEMBL2164509)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetGrowth hormone secretagogue receptor type 1(Human)
Sanofi Research

Curated by ChEMBL
LigandPNGBDBM50395760(CHEMBL2164510)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human GHSR1 expressed in CHO-CREluc cells after 4 hrs by Luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed