Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50040339
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392849(CHEMBL2151190 | US9073941, 612)
Affinity DataIC50:  500nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392855(CHEMBL1969923)
Affinity DataIC50:  630nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392849(CHEMBL2151190 | US9073941, 612)
Affinity DataIC50:  700nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392849(CHEMBL2151190 | US9073941, 612)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392855(CHEMBL1969923)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392856(CHEMBL1981814)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392856(CHEMBL1981814)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392850(CHEMBL2151191)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392852(CHEMBL2151193)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392854(CHEMBL1980140)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392850(CHEMBL2151191)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392851(CHEMBL2151192)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392852(CHEMBL2151193)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392857(CHEMBL1492532)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392860(CHEMBL2151286)
Affinity DataIC50:  7.80E+3nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392853(CHEMBL2000337)
Affinity DataIC50:  1.07E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392858(FURALTADONE)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392851(CHEMBL2151192)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392859(CHEMBL2151285)
Affinity DataIC50:  1.45E+4nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392860(CHEMBL2151286)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392859(CHEMBL2151285)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392852(CHEMBL2151193)
Affinity DataIC50:  2.15E+4nMAssay Description:Inhibition of human JNK2alpha2 using GST-c-jun (1 to 221) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392852(CHEMBL2151193)
Affinity DataIC50:  4.10E+4nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392853(CHEMBL2000337)
Affinity DataIC50:  4.30E+4nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392853(CHEMBL2000337)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392851(CHEMBL2151192)
Affinity DataIC50:  5.80E+4nMAssay Description:Displacement of FITC-JIP peptide from human His-tagged JNK2alpha2 after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392851(CHEMBL2151192)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392853(CHEMBL2000337)
Affinity DataIC50:  1.97E+5nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392850(CHEMBL2151191)
Affinity DataIC50:  2.52E+5nMAssay Description:Inhibition of p38MAPKalpha using GST-ATF2 (1 to 115) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 1(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50392850(CHEMBL2151191)
Affinity DataIC50:  2.95E+5nMAssay Description:Inhibition of rat ERK2 using Ets1 (1 to 138) as substrate preincubated for 30 mins before [gamma-32P]-ATP addition measured after 10 mins by liquid s...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed