Compile Data Set for Download or QSAR
Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50042846
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432146BDBM50432146(CHEMBL2346788)
Affinity DataEC50:  60nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432113BDBM50432113(CHEMBL2349575)
Affinity DataEC50:  60nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432119BDBM50432119(CHEMBL2349603)
Affinity DataEC50:  60nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50416875BDBM50416875(CINACALCET | AMG-073 | AMG073 HCL | CINACALCET HYD...)
Affinity DataEC50:  80nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50299670BDBM50299670((R)-3-(2-chlorophenyl)-N-(1-(3-methoxyphenyl)ethyl...)
Affinity DataEC50:  80nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432145BDBM50432145(CHEMBL2349577)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432148BDBM50432148(CHEMBL2346786)
Affinity DataEC50:  100nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432132BDBM50432132(CHEMBL2349590)
Affinity DataEC50:  130nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432138BDBM50432138(CHEMBL2349584)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432120BDBM50432120(CHEMBL2349602)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432136BDBM50432136(CHEMBL2349586)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432142BDBM50432142(CHEMBL2349580)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432115BDBM50432115(CHEMBL2349573)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432147BDBM50432147(CHEMBL2346787)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432118BDBM50432118(CHEMBL2349604)
Affinity DataEC50:  150nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432122BDBM50432122(CHEMBL2349600)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432121BDBM50432121(CHEMBL2349601)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432127BDBM50432127(CHEMBL2349595)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432141BDBM50432141(CHEMBL2349581)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432112BDBM50432112(CHEMBL2349576)
Affinity DataEC50:  200nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432123BDBM50432123(CHEMBL2349599)
Affinity DataEC50:  300nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432139BDBM50432139(CHEMBL2349583)
Affinity DataEC50:  300nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432124BDBM50432124(CHEMBL2349598)
Affinity DataEC50:  300nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432117BDBM50432117(CHEMBL2349605)
Affinity DataEC50:  300nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432131BDBM50432131(CHEMBL2349591)
Affinity DataEC50:  350nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432137BDBM50432137(CHEMBL2349585)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432125BDBM50432125(CHEMBL2349597)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432128BDBM50432128(CHEMBL2349594)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432144BDBM50432144(CHEMBL2349578)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432133BDBM50432133(CHEMBL2349589)
Affinity DataEC50:  400nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432135BDBM50432135(CHEMBL2349587)
Affinity DataEC50:  550nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432116BDBM50432116(CHEMBL2346765)
Affinity DataEC50:  600nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432126BDBM50432126(CHEMBL2349596)
Affinity DataEC50:  800nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432130BDBM50432130(CHEMBL2349592)
Affinity DataEC50:  800nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432134BDBM50432134(CHEMBL2349588)
Affinity DataEC50:  800nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432150BDBM50432150(CHEMBL2346784)
Affinity DataEC50:  800nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 61401BDBM61401(FENDILINE HYDROCHLORIDE | MLS000069570 | CHEMBL254...)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432140BDBM50432140(CHEMBL2349582)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432114BDBM50432114(CHEMBL2349574)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432129BDBM50432129(CHEMBL2349593)
Affinity DataEC50:  1.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432152BDBM50432152(CHEMBL2346782)
Affinity DataEC50:  1.50E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432143BDBM50432143(CHEMBL2349579)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432159BDBM50432159(CHEMBL2346776)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432151BDBM50432151(CHEMBL2346783)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432164BDBM50432164(CHEMBL2346771)
Affinity DataEC50:  2.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432158BDBM50432158(CHEMBL2346777)
Affinity DataEC50:  3.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432163BDBM50432163(CHEMBL2346772)
Affinity DataEC50:  3.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432154BDBM50432154(CHEMBL2346780)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432162BDBM50432162(1-(3,3-diphenylpropyl)-3-p-tolylurea | CHEMBL23467...)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetExtracellular calcium-sensing receptor(Human)
Galapagos

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50432161BDBM50432161(CHEMBL2346774)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive allosteric modulation of human CaSR transfected in CHO cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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