TargetPlasma kallikrein(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Inhibition of human recombinant polyhistidine-tagged plasma kallikrein expressed in Escherichia coli XL1 blue using Z-FR-AMC as substrate by fluorime...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 3.10E+3nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 3.30E+3nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 4.70E+3nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 5.00E+3nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 7.80E+3nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 8.30E+3nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 8.30E+3nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 1.02E+4nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 1.12E+4nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 1.42E+4nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 2.05E+4nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 3.35E+4nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >7.50E+4nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetCoagulation factor XII(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >7.50E+4nMAssay Description:Inhibition of human biotinylated beta factor 12a expressed in Escherichia coli TG1 using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: 1.18E+5nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasma kallikrein(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human PK using Z-Phe-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human thrombin using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetSerine protease 1(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human trypsin using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetSerine protease 1(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human trypsin using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human plasmin using H-D-Val-Leu-Lys-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetProthrombin(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human thrombin using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity by fluorescence plate reader analysisMore data for this Ligand-Target Pair
TargetPlasma kallikrein(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human PK using Z-Phe-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human coagulation factor 11a using Boc-Phe-Ser-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human uPA using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human tPA using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human tPA using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human uPA using Z-Gly-Gly-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair
TargetCoagulation factor XI(Homo sapiens (Human))
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Ecole Polytechnique F�D�Rale De Lausanne Epfl
Curated by ChEMBL
Affinity DataKi: >1.20E+5nMAssay Description:Inhibition of human coagulation factor 11a using Boc-Phe-Ser-Arg-AMC as substrate assessed as residual activity by fluorometric analysisMore data for this Ligand-Target Pair