Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50005596
TargetSodium channel protein type 2 subunit alpha(Rattus norvegicus)
Institute Of Nuclear Medicine

Curated by ChEMBL
LigandPNGBDBM50030510(CHEMBL299668 | [1-Benzyl-7-chloro-1H-quinolin-(4E)...)
Affinity DataKi:  9nMAssay Description:Inhibition of rat brain voltage-gated sodium channel subunit alpha Nav1.2-mediated current expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Institute Of Nuclear Medicine

Curated by ChEMBL
LigandPNGBDBM50493060(CHEMBL2419774)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human voltage-gated sodium channel subunit alpha Nav1.2 expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 2 subunit alpha(Homo sapiens (Human))
Institute Of Nuclear Medicine

Curated by ChEMBL
LigandPNGBDBM50030510(CHEMBL299668 | [1-Benzyl-7-chloro-1H-quinolin-(4E)...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human voltage-gated sodium channel subunit alpha Nav1.2 expressed in CHO cells by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed