Compile Data Set for Download or QSAR
maximum 50k data
Found 60 Enz. Inhib. hit(s) with all data for entry = 50005920
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126727((S)-4-(3-(4-(4-fluorophenyl)piperazin-1-yl)-2-(N-m...)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404086(CHEMBL341226)
Affinity DataIC50:  5nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126702(CHEMBL282807 | Isoquinoline-5-sulfonic acid 4-{(S)...)
Affinity DataIC50:  5.80nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126713(CHEMBL282173 | Isoquinoline-5-sulfonic acid 4-{(S)...)
Affinity DataIC50:  5.80nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404085(CHEMBL336619)
Affinity DataIC50:  7.90nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50411888(CHEMBL270421)
Affinity DataIC50:  9.10nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404090(CHEMBL424451)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415889(CHEMBL1098723)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126715(CHEMBL27837 | Isoquinoline-5-sulfonic acid 4-[(S)-...)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126723((S)-4-(3-(4-(3-chlorophenyl)piperazin-1-yl)-2-(N-m...)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126718((S)-4-(3-(4-(2-chlorophenyl)piperazin-1-yl)-2-(N-m...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423270(CHEMBL393241)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415882(CHEMBL1094106)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415908(CHEMBL1094641)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423276(CHEMBL396587)
Affinity DataIC50:  27nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126712(CHEMBL27711 | Isoquinoline-5-sulfonic acid 4-{(S)-...)
Affinity DataIC50:  34nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50410952(CHEMBL208560)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423280(CHEMBL245561)
Affinity DataIC50:  49nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415888(CHEMBL1096314)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423272(CHEMBL246578)
Affinity DataIC50:  50nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415891(CHEMBL1094744)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50495434(CHEMBL131241)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126719((S)-4-(3-(4-benzylpiperazin-1-yl)-2-(N-methylisoqu...)
Affinity DataIC50:  65nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126724(CHEMBL282808 | Isoquinoline-5-sulfonic acid 4-{(S)...)
Affinity DataIC50:  71nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50411878(CHEMBL245754)
Affinity DataIC50:  78nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415909(CHEMBL1094482)
Affinity DataIC50:  79nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50087267((1-(N,O-bis(1,5-isoquinolinesulfonyl)-N-methyl-L-t...)
Affinity DataIC50:  94nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126717(CHEMBL286496 | Isoquinoline-5-sulfonic acid 4-{(S)...)
Affinity DataIC50:  98nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126710(CHEMBL28152 | Isoquinoline-5-sulfonic acid 4-{(S)-...)
Affinity DataIC50:  101nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126706((S)-4-(3-(4-(4-chlorophenyl)piperazin-1-yl)-2-(N-m...)
Affinity DataIC50:  105nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415906(CHEMBL1096096)
Affinity DataIC50:  126nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404074(CHEMBL337873)
Affinity DataIC50:  126nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126711(CHEMBL28374 | Isoquinoline-5-sulfonic acid 4-{(S)-...)
Affinity DataIC50:  132nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415898(CHEMBL1096100)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415884(CHEMBL1096049)
Affinity DataIC50:  158nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50126709(CHEMBL27106 | Isoquinoline-5-sulfonic acid 4-{(S)-...)
Affinity DataIC50:  176nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423269(CHEMBL245755)
Affinity DataIC50:  191nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415913(CHEMBL1096048)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423282(CHEMBL246770)
Affinity DataIC50:  209nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50423277(CHEMBL245578)
Affinity DataIC50:  214nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50495436(CHEMBL3108814)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415885(CHEMBL1096660)
Affinity DataIC50:  316nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50404076(CHEMBL337419)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50495438(CHEMBL3108810)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50495437(CHEMBL3108813)
Affinity DataIC50:  501nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415893(CHEMBL1095395)
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415899(CHEMBL1096099)
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415896(CHEMBL1096030)
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415903(CHEMBL1094485)
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 7(Homo sapiens (Human))
Punjabi University

Curated by ChEMBL
LigandPNGBDBM50415900(CHEMBL1095783)
Affinity DataIC50: <1.00E+3nMAssay Description:Antagonist activity at P2X7 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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