Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 7990
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM227598(Penem 1)
Affinity DataKi:  30nM IC50: 150nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2017
Entry Details Article
PubMed
TargetBeta-lactamase OXA-1(Escherichia coli)
Case Western Reserve University

LigandPNGBDBM227598(Penem 1)
Affinity DataKi:  50nM IC50: 30nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2017
Entry Details Article
PubMed
TargetBeta-lactamase OXA-1(Escherichia coli)
Case Western Reserve University

LigandPNGBDBM227599(Penem 3)
Affinity DataKi:  380nM IC50: 60nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2017
Entry Details Article
PubMed
TargetOxa40(Acinetobacter baumannii)
Case Western Reserve University

LigandPNGBDBM227599(Penem 3)
Affinity DataKi:  150nM IC50: 160nMpH: 7.2Assay Description:Steady-state kinetics were performed on an Agilent 8453 diode array spectrophotometer (Palo Alto, CA) in 50 mM sodium phosphate buffer (pH 7.2) suppl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2017
Entry Details Article
PubMed