Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50040352
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393034(CHEMBL2152704)
Affinity DataIC50:  160nMAssay Description:Inhibition of EphB4 in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393034(CHEMBL2152704)
Affinity DataIC50:  300nMAssay Description:Inhibition of EphB4 by FRET assay in presence of 30 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393034(CHEMBL2152704)
Affinity DataIC50:  338nMAssay Description:Inhibition of recombinant Src catalytic domain in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393034(CHEMBL2152704)
Affinity DataIC50:  864nMAssay Description:Inhibition of recombinant Abl1 catalytic domain in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393034(CHEMBL2152704)
Affinity DataIC50:  930nMAssay Description:Inhibition of human full length EphB4 expressed in MEF cells assessed as inhibition of human ephrin B2/FC chimera-stimulated receptor autophosphoryla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393034(CHEMBL2152704)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of recombinant Lck catalytic domain in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393034(CHEMBL2152704)
Affinity DataIC50:  1.62E+3nMAssay Description:Inhibition of recombinant EGFR catalytic domain in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393033(CHEMBL2152699)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of EphB4 in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393035(CHEMBL2152698)
Affinity DataIC50:  8.40E+3nMAssay Description:Inhibition of EphB4 in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393033(CHEMBL2152699)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of EphB4 by FRET assay in presence of 30 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEphrin type-B receptor 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50393036(CHEMBL2152702)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of EphB4 in presence of 1 uM radiolabeled ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed