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Found 26 Enz. Inhib. hit(s) with all data for entry = 50045165
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048063(CHEMBL3314943)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438783(CHEMBL2415106)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048063(CHEMBL3314943)
Affinity DataKi:  1.21E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438783(CHEMBL2415106)
Affinity DataKi:  4.11E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048065(CHEMBL3314941)
Affinity DataKi:  8.60E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438782(CHEMBL2413162)
Affinity DataKi:  8.67E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438779(CHEMBL2413161)
Affinity DataKi:  8.88E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048065(CHEMBL3314941)
Affinity DataKi:  9.18E+3nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048064(CHEMBL3314942)
Affinity DataKi: >2.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB1 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048064(CHEMBL3314942)
Affinity DataKi:  2.26E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438779(CHEMBL2413161)
Affinity DataKi:  4.40E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438782(CHEMBL2413162)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]CP55,940 from human CB2 expressed in CHO-K1 cells after 2 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438783(CHEMBL2415106)
Affinity DataIC50:  4.07E+3nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50107607((5Z,8Z)-Icosa-5,8,11,14-tetraenoic acid (furan-3-y...)
Affinity DataIC50:  7.24E+3nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438779(CHEMBL2413161)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048064(CHEMBL3314942)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048065(CHEMBL3314941)
Affinity DataIC50:  1.78E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438782(CHEMBL2413162)
Affinity DataIC50:  1.91E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048063(CHEMBL3314943)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048066(CHEMBL1316265 | OMDM2 | US10300048, Compound OMDM-...)
Affinity DataIC50:  2.33E+4nMAssay Description:Inhibition of FAAH-mediated [ethanol-amine-1-3H]AEA hydrolysis in human U937 cells preincubated for 15 mins measured 15 mins post AEA addition by liq...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Mus musculus (mouse))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438783(CHEMBL2415106)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Mus musculus (mouse))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048063(CHEMBL3314943)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Mus musculus (mouse))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438782(CHEMBL2413162)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Mus musculus (mouse))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048065(CHEMBL3314941)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Mus musculus (mouse))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50048064(CHEMBL3314942)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Mus musculus (mouse))
University Of Szeged

Curated by ChEMBL
LigandPNGBDBM50438779(CHEMBL2413161)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of mouse brain MAGL-mediated [glycerol-1,2,3-3H]-2-OG hydrolysis preincubated for 15 mins measured 15 mins post 2-OG addition by liquid sc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed