Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 6309
TargetMitogen-activated protein kinase 1(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 2.70nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 8.30nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 104nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase 17A(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 114nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase TTK(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 193nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 3(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataKd:  213nMpH: 7.5 T: 2°CAssay Description:For ERK1 and ERK2, the buffer contained 20 mM HEPES (pH 7.5), 150 mM NaCl and 0.5 mM TCEP. For haspin, the buffer contained 20 mM HEPES (pH 7.5), 250...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataKd:  233nMpH: 7.5 T: 2°CAssay Description:For ERK1 and ERK2, the buffer contained 20 mM HEPES (pH 7.5), 150 mM NaCl and 0.5 mM TCEP. For haspin, the buffer contained 20 mM HEPES (pH 7.5), 250...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin [465-798](Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataKd:  297nMpH: 7.5 T: 2°CAssay Description:For ERK1 and ERK2, the buffer contained 20 mM HEPES (pH 7.5), 150 mM NaCl and 0.5 mM TCEP. For haspin, the buffer contained 20 mM HEPES (pH 7.5), 250...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 1(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataKd:  300nMpH: 7.5 T: 2°CAssay Description:For ERK1 and ERK2, the buffer contained 20 mM HEPES (pH 7.5), 150 mM NaCl and 0.5 mM TCEP. For haspin, the buffer contained 20 mM HEPES (pH 7.5), 250...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 3(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 304nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase haspin [465-798](Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 398nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 4(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 503nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 508nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase D1(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 535nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetAurora kinase C(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 580nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 632nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 783nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMisshapen-like kinase 1(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 942nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8 [1-363](Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 1.08E+3nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha'(Human)
George Washington University

LigandPNGBDBM103302(SCH772984 | US8546404, 6)
Affinity DataIC50: 1.00E+4nMAssay Description:The IC50 values of selected kinases were determined using either Z'LYTE, Adapta or LanthaScreen assays.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2014
Entry Details Article
PubMed