Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50045028
TargetAmine oxidase [flavin-containing] B(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50042275(CHEMBL3360732)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50042280(CHEMBL3360734)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50042281(CHEMBL3360735)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50042277(CHEMBL3360731)
Affinity DataIC50: 6nMAssay Description:Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 20nMAssay Description:Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM15613(MCL | Aurorix | 4-chloro-N-[2-(morpholin-4-yl)ethy...)
Affinity DataIC50: 361nMAssay Description:Inhibition of human recombinant MAOA expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50042279(CHEMBL3360733)
Affinity DataIC50: 2.17E+3nMAssay Description:Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50042275(CHEMBL3360732)
Affinity DataIC50: 4.18E+3nMAssay Description:Inhibition of human recombinant MAOA expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50042276(CHEMBL3360730)
Affinity DataIC50: 5.52E+3nMAssay Description:Inhibition of human recombinant MAOB expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Human)
Universidad De Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 6.72E+4nMAssay Description:Inhibition of human recombinant MAOA expressed in BTI-TN-5B1-4 cells using p-tyramine substrate assessed as reduction in H2O2 productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2016
Entry Details Article
PubMed