Compile Data Set for Download or QSAR
Report error Found 74 Enz. Inhib. hit(s) with all data for entry = 50046079
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093793BDBM50093793(E-2006 | Lemborexant)
Affinity DataKi:  0.440nMAssay Description:Binding affinity to human OX2R expressed in HEK-293 cells assessed as inhibition of orexin A-induced calcium accumulation by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093815BDBM50093815(CHEMBL3585948)
Affinity DataKi:  2nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093788BDBM50093788(CHEMBL3585957)
Affinity DataKi:  2nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093791BDBM50093791(CHEMBL3585955)
Affinity DataKi:  3nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093793BDBM50093793(E-2006 | Lemborexant)
Affinity DataKi:  3nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093795BDBM50093795(CHEMBL3585952)
Affinity DataKi:  3nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093788BDBM50093788(CHEMBL3585957)
Affinity DataKi:  4nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093790BDBM50093790(CHEMBL3585956)
Affinity DataKi:  4nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093798BDBM50093798(CHEMBL3585951)
Affinity DataKi:  4nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029064BDBM50029064(CHEMBL3343259)
Affinity DataKi:  5nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093793BDBM50093793(E-2006 | Lemborexant)
Affinity DataKi:  5.70nMAssay Description:Binding affinity to human OX1R expressed in HEK-293 cells assessed as inhibition of orexin A-induced calcium accumulation by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093793BDBM50093793(E-2006 | Lemborexant)
Affinity DataKi:  6nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093798BDBM50093798(CHEMBL3585951)
Affinity DataKi:  6nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093795BDBM50093795(CHEMBL3585952)
Affinity DataKi:  6nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093900BDBM50093900(CHEMBL3585946)
Affinity DataKi:  7nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093791BDBM50093791(CHEMBL3585955)
Affinity DataKi:  7nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094022BDBM50094022(CHEMBL3585940)
Affinity DataKi:  7nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094039BDBM50094039(CHEMBL3585938)
Affinity DataKi:  8nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093792BDBM50093792(CHEMBL3585954)
Affinity DataKi:  8nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094006BDBM50094006(CHEMBL3585942)
Affinity DataKi:  9nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093780BDBM50093780(CHEMBL3585936)
Affinity DataKi:  10nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093790BDBM50093790(CHEMBL3585956)
Affinity DataKi:  14nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093794BDBM50093794(CHEMBL3585953)
Affinity DataKi:  17nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094007BDBM50094007(CHEMBL3585941)
Affinity DataKi:  21nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093800BDBM50093800(CHEMBL3585950)
Affinity DataKi:  29nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093801BDBM50093801(CHEMBL3585949)
Affinity DataKi:  34nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093815BDBM50093815(CHEMBL3585948)
Affinity DataKi:  39nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093792BDBM50093792(CHEMBL3585954)
Affinity DataKi:  39nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094006BDBM50094006(CHEMBL3585942)
Affinity DataKi:  43nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094038BDBM50094038(CHEMBL3585939)
Affinity DataKi:  49nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093976BDBM50093976(CHEMBL3585944)
Affinity DataKi:  50nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093897BDBM50093897(CHEMBL3585947)
Affinity DataKi:  56nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094007BDBM50094007(CHEMBL3585941)
Affinity DataKi:  73nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094005BDBM50094005(CHEMBL3585943)
Affinity DataKi:  80nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093794BDBM50093794(CHEMBL3585953)
Affinity DataKi:  81nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50029064BDBM50029064(CHEMBL3343259)
Affinity DataKi:  106nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094022BDBM50094022(CHEMBL3585940)
Affinity DataKi:  121nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093801BDBM50093801(CHEMBL3585949)
Affinity DataKi:  124nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093900BDBM50093900(CHEMBL3585946)
Affinity DataKi:  137nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093897BDBM50093897(CHEMBL3585947)
Affinity DataKi:  138nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093975BDBM50093975(CHEMBL3585945)
Affinity DataKi:  163nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094039BDBM50094039(CHEMBL3585938)
Affinity DataKi:  171nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093782BDBM50093782(CHEMBL3585935)
Affinity DataKi:  204nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin receptor type 2(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093787BDBM50093787(CHEMBL3585933)
Affinity DataKi:  222nMAssay Description:Binding affinity to human OX2R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093800BDBM50093800(CHEMBL3585950)
Affinity DataKi:  224nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093780BDBM50093780(CHEMBL3585936)
Affinity DataKi:  391nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093976BDBM50093976(CHEMBL3585944)
Affinity DataKi:  391nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093787BDBM50093787(CHEMBL3585933)
Affinity DataKi:  938nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50094005BDBM50094005(CHEMBL3585943)
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
TargetOrexin/Hypocretin receptor type 1(Human)
Eisai

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50093975BDBM50093975(CHEMBL3585945)
Affinity DataKi:  1.58E+3nMAssay Description:Binding affinity to human OX1R by radioligand displacement binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2016
Entry Details Article
PubMed
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