TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant GST-fused Dyrk2 expressed in Escherichia coli using Woodtide as substrate after 15 mins by P81 membrane assay in pres...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of human recombinant Dyrk1B using Woodtide as substrate after 15 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of Dyrk1A (unknown origin) using dynatide 3 as substrate after 10 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant His6-tagged Dyrk1A expressed in Escherichia coli using Woodtide as substrate after 15 mins by P81 membrane assay in p...More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of Dyrk1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(RAT)
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 330nMAssay Description:Inhibition of rat Dyrk1A using Woodtide as substrate after 40 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:Inhibition of Dyrk1A (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of Dyrk2 (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of Dyrk3 (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
India Academy Of Scientific & Innovative Research (Acsir)
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of Dyrk1A (unknown origin) using Woodtide as substrate after 30 mins by P81 membrane assay in presence of [33P]-g-ATPMore data for this Ligand-Target Pair