Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 50046845
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134199(CHEMBL3735057)
Affinity DataKi:  627nMAssay Description:Displacement of [3H]furoyl-LIGRL-NH2 from human protease-activated receptor 2 in NCTC-2544 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134200(CHEMBL3735405)
Affinity DataKi:  1.94E+3nMAssay Description:Displacement of [3H]furoyl-LIGRL-NH2 from human protease-activated receptor 2 in NCTC-2544 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134198(CHEMBL1684609)
Affinity DataIC50:  690nMAssay Description:Antagonist activity at protease-activated receptor 2 (unknown origin) expressed in CHO-K1 cells assessed as inhibition of trypsin-induced calcium flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50440868(CHEMBL2431617)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at protease-activated receptor 2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134197(CHEMBL3735493)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at protease-activated receptor 2 (unknown origin) expressed in CHO-K1 cells assessed as inhibition of trypsin-induced calcium flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134196(CHEMBL3736126)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at protease-activated receptor 2 (unknown origin) expressed in CHO-K1 cells assessed as inhibition of trypsin-induced calcium flu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50134201(CHEMBL3734977)
Affinity DataIC50:  5.00E+6nMAssay Description:Displacement of [3H]furoyl-LIGRL-NH2 from human protease-activated receptor 2 in NCTC-2544 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed