Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 50047283
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157618BDBM50157618(CHEMBL3785637)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157618BDBM50157618(CHEMBL3785637)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157617BDBM50157617(CHEMBL3785764)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157619BDBM50157619(CHEMBL3787072)
Affinity DataEC50:  48nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157615BDBM50157615(CHEMBL3787463)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157614BDBM50157614(CHEMBL3786972)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275510BDBM50275510(3-(4-(Phenylethynyl)phenyl)propanoic acid | CHEMBL...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157603BDBM50157603(CHEMBL3786524)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157616BDBM50157616(CHEMBL3786526)
Affinity DataEC50:  209nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157568BDBM50157568(CHEMBL3787580)
Affinity DataEC50:  389nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157613BDBM50157613(CHEMBL3785544)
Affinity DataEC50:  417nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157620BDBM50157620(CHEMBL3785413)
Affinity DataEC50:  427nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157600BDBM50157600(CHEMBL3787110)
Affinity DataEC50:  490nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157601BDBM50157601(CHEMBL3786418)
Affinity DataEC50:  513nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157567BDBM50157567(CHEMBL3785789)
Affinity DataEC50:  1.45E+3nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157569BDBM50157569(CHEMBL3787151)
Affinity DataEC50:  1.82E+3nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240347BDBM50240347((Z,Z,Z)-9,12,15-octadecatrienoic acid | cis,cis,ci...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50240347BDBM50240347((Z,Z,Z)-9,12,15-octadecatrienoic acid | cis,cis,ci...)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157567BDBM50157567(CHEMBL3785789)
Affinity DataEC50:  4.07E+3nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157569BDBM50157569(CHEMBL3787151)
Affinity DataEC50:  4.79E+3nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157571BDBM50157571(CHEMBL3786964)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157614BDBM50157614(CHEMBL3786972)
Affinity DataEC50:  7.59E+3nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50275510BDBM50275510(3-(4-(Phenylethynyl)phenyl)propanoic acid | CHEMBL...)
Affinity DataEC50:  8.51E+3nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157601BDBM50157601(CHEMBL3786418)
Affinity DataEC50:  9.55E+3nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157568BDBM50157568(CHEMBL3787580)
Affinity DataEC50:  1.05E+4nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157619BDBM50157619(CHEMBL3787072)
Affinity DataEC50:  1.78E+4nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157618BDBM50157618(CHEMBL3785637)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157617BDBM50157617(CHEMBL3785764)
Affinity DataEC50:  2.63E+4nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157600BDBM50157600(CHEMBL3787110)
Affinity DataEC50:  3.39E+4nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157616BDBM50157616(CHEMBL3786526)
Affinity DataEC50:  3.47E+4nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157615BDBM50157615(CHEMBL3787463)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157566BDBM50157566(CHEMBL3785667)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157613BDBM50157613(CHEMBL3785544)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157566BDBM50157566(CHEMBL3785667)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157620BDBM50157620(CHEMBL3785413)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 1(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157602BDBM50157602(CHEMBL3787165)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human FFA1 receptor expressed in human 1321N1 cells measured for 50 intervals of 0.4 secs by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157571BDBM50157571(CHEMBL3786964)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157602BDBM50157602(CHEMBL3787165)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed
TargetFree fatty acid receptor 4(Human)
University of Southern Denmark

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50157603BDBM50157603(CHEMBL3786524)
Affinity DataEC50: <1.00E+5nMAssay Description:Agonist activity at human C-terminal YFP-tagged FFA4 receptor expressed in HEK293 cells incubated for 5 mins by BRET based beta-arrestin 2 recruitmen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2017
Entry Details Article
PubMed