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Found 30 Enz. Inhib. hit(s) with all data for entry = 50047501
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM10246((4S)-4-{[(1S)-1-{[(2S)-1-carboxy-3-oxopropan-2-yl]...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM10246((4S)-4-{[(1S)-1-{[(2S)-1-carboxy-3-oxopropan-2-yl]...)
Affinity DataIC50:  60nMAssay Description:Inhibition of His-tagged human recombinant caspase 7 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171526(CHEMBL3805744)
Affinity DataIC50:  1.94E+4nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171527(CHEMBL3806315)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171506(CHEMBL3805942)
Affinity DataIC50:  3.72E+4nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171528(CHEMBL3806289)
Affinity DataIC50:  3.83E+4nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171505(CHEMBL3805088)
Affinity DataIC50:  5.23E+4nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171507(CHEMBL3805488)
Affinity DataIC50:  6.32E+4nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171508(CHEMBL3805483)
Affinity DataIC50:  1.22E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171509(CHEMBL3805916)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171510(CHEMBL3805458)
Affinity DataIC50:  1.32E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171533(CHEMBL3805517)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 7 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171563(CHEMBL3805045)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 7 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171564(CHEMBL3805555)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 7 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171532(CHEMBL3805972)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 7 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171526(CHEMBL3805744)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 7 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171506(CHEMBL3805942)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 7 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-7(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171503(CHEMBL3805109)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 7 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171501(CHEMBL3805231)
Affinity DataIC50:  2.02E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171502(CHEMBL3804942)
Affinity DataIC50:  2.78E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171503(CHEMBL3805109)
Affinity DataIC50:  2.97E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171530(CHEMBL3805593)
Affinity DataIC50:  3.10E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171531(CHEMBL3805833)
Affinity DataIC50:  3.51E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171529(CHEMBL3806253)
Affinity DataIC50:  3.75E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171500(CHEMBL3805818)
Affinity DataIC50:  4.56E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171532(CHEMBL3805972)
Affinity DataIC50:  4.87E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171533(CHEMBL3805517)
Affinity DataIC50:  5.47E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171563(CHEMBL3805045)
Affinity DataIC50:  5.52E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171564(CHEMBL3805555)
Affinity DataIC50:  5.99E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
The Fifth Affiliated Hospital Of Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50171565(CHEMBL3805679)
Affinity DataIC50:  6.74E+5nMAssay Description:Inhibition of His-tagged human recombinant caspase 3 expressed in Escherichia coli using acetyl-Asp-Glu-Val-Asp-7- amido-4-methylcoumarin (Ac-DEVD-AM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed