Compile Data Set for Download or QSAR
Report error Found 212 Enz. Inhib. hit(s) with all data for entry = 50009826
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 1 hr by liquid scintillation spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50180036(CHEMBL371214 | (6aR,10aR)-3-(1,1-dimethylbutyl)-6a...)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 1 hr by liquid scintillation spectrometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532455(CHEMBL4557358)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532455(CHEMBL4557358)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataIC50: 4.20nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataIC50: 4.20nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532460(CHEMBL4441538)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532460(CHEMBL4441538)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532476(CHEMBL4527391)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532476(CHEMBL4527391)
Affinity DataKi:  5.20nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataIC50: 8.30nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataIC50: 8.30nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532454(CHEMBL4588694)
Affinity DataIC50: 14nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532467(CHEMBL4467761)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532467(CHEMBL4467761)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532454(CHEMBL4588694)
Affinity DataIC50: 14nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532438(CHEMBL4441649)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532479(CHEMBL4463214)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532479(CHEMBL4463214)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532438(CHEMBL4441649)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532455(CHEMBL4557358)
Affinity DataIC50: 22nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532455(CHEMBL4557358)
Affinity DataIC50: 22nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532474(CHEMBL4465748)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532474(CHEMBL4465748)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50265621(HU-308 | ((1R,4S,5R)-4-(2,6-dimethoxy-4-(2-methylo...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]HU-243 from rat CB2 receptor expressed in African green monkey COS7 cell membranes after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Rat)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50265621(HU-308 | ((1R,4S,5R)-4-(2,6-dimethoxy-4-(2-methylo...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]HU-243 from rat CB2 receptor expressed in African green monkey COS7 cell membranes after 90 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532443(CHEMBL4441832)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532443(CHEMBL4441832)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532453(CHEMBL4562832)
Affinity DataIC50: 26nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532453(CHEMBL4562832)
Affinity DataIC50: 26nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532461(CHEMBL4472364)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532461(CHEMBL4472364)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-CP55940 from human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532456(CHEMBL4581919)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532448(CHEMBL4475298)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532456(CHEMBL4581919)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532448(CHEMBL4475298)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-CP55940 from human CB2 receptor expressed in HEK293 cell membranes after 90 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
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