Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50047792
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190152(CHEMBL3827259)
Affinity DataIC50:  7.5nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190168(CHEMBL3827304)
Affinity DataIC50:  9.60nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190151(CHEMBL3827570)
Affinity DataIC50:  18nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190148(CHEMBL3828187)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190155(CHEMBL3827736)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190162(CHEMBL3827475)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190153(CHEMBL3828483)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190149(CHEMBL3827041)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190166(CHEMBL3827830)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190150(CHEMBL3827209)
Affinity DataIC50:  39nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190156(CHEMBL3828154)
Affinity DataIC50:  46nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190165(CHEMBL3827577)
Affinity DataIC50:  51nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190158(CHEMBL3827154)
Affinity DataIC50:  59nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190154(CHEMBL3827723)
Affinity DataIC50:  64nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190159(CHEMBL3827356)
Affinity DataIC50:  77nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190157(CHEMBL3827912)
Affinity DataIC50:  117nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190160(CHEMBL3828182)
Affinity DataIC50:  203nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190161(CHEMBL3827410)
Affinity DataIC50:  457nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190164(CHEMBL3827473)
Affinity DataIC50:  489nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190163(CHEMBL3828329)
Affinity DataIC50:  1.33E+3nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50190167(CHEMBL3827898)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at calcium sensing receptor (unknown origin) by cell based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed