Compile Data Set for Download or QSAR
Report error Found 62 Enz. Inhib. hit(s) with all data for entry = 50018883
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50030448(CHEMBL269732 | 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN ...)
Affinity DataKd:  0.400nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM36609(Rapamycin C-7, analog 4 | SIROLIMUS | US11603377, ...)
Affinity DataKd:  3.70nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613636(CHEMBL5286207)
Affinity DataKi:  4nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM36609(Rapamycin C-7, analog 4 | SIROLIMUS | US11603377, ...)
Affinity DataKd:  4.20nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKd:  6nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613631(CHEMBL5281156)
Affinity DataKi:  6nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613624(CHEMBL5291300)
Affinity DataKi:  7nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM23334(3-(pyridin-3-yl)propyl (2S)-1-(3,3-dimethyl-2-oxop...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50116636(1-(3,3-Dimethyl-2-oxo-pentanoyl)-pyrrolidine-2-car...)
Affinity DataKi:  11nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613623(CHEMBL5280097)
Affinity DataKi:  12nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613629(CHEMBL5268140)
Affinity DataIC50: 14nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50132556((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataKi:  20nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613634(CHEMBL5289205)
Affinity DataKi:  23nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50030448(CHEMBL269732 | 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN ...)
Affinity DataKd:  23nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613635(CHEMBL5291024)
Affinity DataKi:  26nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50030448(CHEMBL269732 | 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN ...)
Affinity DataKi:  93nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50030448(CHEMBL269732 | 8-DEETHYL-8-[BUT-3-ENYL]-ASCOMYCIN ...)
Affinity DataKd:  104nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50067006((S)-1-(3,3-Dimethyl-2-oxo-pentanoyl)-piperidine-2-...)
Affinity DataKi:  110nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50381013(CHEMBL2017129)
Affinity DataIC50: 200nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613628(CHEMBL5279925)
Affinity DataIC50: 300nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM92913(Aryl 1-indanylketone, 2)
Affinity DataIC50: 300nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613625(CHEMBL1235853)
Affinity DataKi:  300nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM23334(3-(pyridin-3-yl)propyl (2S)-1-(3,3-dimethyl-2-oxop...)
Affinity DataKi:  306nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM92913(Aryl 1-indanylketone, 2)
Affinity DataIC50: 400nMAssay Description:Inhibition of Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM23334(3-(pyridin-3-yl)propyl (2S)-1-(3,3-dimethyl-2-oxop...)
Affinity DataKi:  447nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50381013(CHEMBL2017129)
Affinity DataIC50: 520nMAssay Description:Inhibition of CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613622(CHEMBL5279437)
Affinity DataKd:  660nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  800nMAssay Description:Binding affinity to Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM23334(3-(pyridin-3-yl)propyl (2S)-1-(3,3-dimethyl-2-oxop...)
Affinity DataKi:  936nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50080534(ethyl (4-{(2R)-2-[(1S,3S,5S)-3,5-dimethyl-2-oxocyc...)
Affinity DataKi:  958nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50080534(ethyl (4-{(2R)-2-[(1S,3S,5S)-3,5-dimethyl-2-oxocyc...)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM92915(Aryl 1-indanylketone, 4)
Affinity DataKi:  1.20E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50080534(ethyl (4-{(2R)-2-[(1S,3S,5S)-3,5-dimethyl-2-oxocyc...)
Affinity DataKi:  1.69E+3nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50495808(CHEMBL1557710)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase B(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM92915(Aryl 1-indanylketone, 4)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to CypB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613630(BETAMETHASONE PHOSPHORIC ACID | CHEBI:68603 | Beta...)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to Pin1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50381013(CHEMBL2017129)
Affinity DataIC50: 2.42E+3nMAssay Description:Inhibition of CypD (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613627(CHEMBL2006156)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613626(CHEMBL5275318)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to CypD (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613626(CHEMBL5275318)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613627(CHEMBL2006156)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50080528(Cycloheximid | 3-((R)-2-((1S,3S,5S)-3,5-dimethyl-2...)
Affinity DataKi:  3.40E+3nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase D(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM92913(Aryl 1-indanylketone, 2)
Affinity DataIC50: 6.28E+3nMAssay Description:Inhibition of CypD (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613621(CHEMBL5268083)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP51 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613621(CHEMBL5268083)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP12 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP4(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613621(CHEMBL5268083)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to FKBP52 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase B(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM92913(Aryl 1-indanylketone, 2)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of CypB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase A(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50495808(CHEMBL1557710)
Affinity DataKi:  2.10E+4nMAssay Description:Binding affinity to CypA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50613633(CHEMBL5271713)
Affinity DataKi:  2.30E+4nMAssay Description:Binding affinity to wild type FKBP51 (unknown origin) by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargetPeptidyl-prolyl cis-trans isomerase-like 1(Human)
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50381013(CHEMBL2017129)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibition of PPIL1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
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