Compile Data Set for Download or QSAR
maximum 50k data
Found 61 Enz. Inhib. hit(s) with all data for entry = 50010066
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534898(CHEMBL4522563)
Affinity DataIC50:  1nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534903(CHEMBL4580709)
Affinity DataIC50:  2nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50389939(CHEMBL1553629)
Affinity DataIC50:  2nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534869(CHEMBL4474264)
Affinity DataIC50:  2nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534887(CHEMBL4457926)
Affinity DataIC50:  3nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534858(CHEMBL4554003)
Affinity DataIC50:  3nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534892(CHEMBL4436256)
Affinity DataIC50:  3nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534890(CHEMBL4438146)
Affinity DataIC50:  3nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534862(CHEMBL4462538)
Affinity DataIC50:  4nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534860(CHEMBL4449492)
Affinity DataIC50:  4nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534902(CHEMBL4571226)
Affinity DataIC50:  4nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534899(CHEMBL4550424)
Affinity DataIC50:  4nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534867(CHEMBL4447746)
Affinity DataIC50:  5nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534895(CHEMBL4569725)
Affinity DataIC50:  5nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534868(CHEMBL4476181)
Affinity DataIC50:  6nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534910(CHEMBL4521762)
Affinity DataIC50:  7nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534857(CHEMBL4516158)
Affinity DataIC50:  8nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534870(CHEMBL4589557)
Affinity DataIC50:  8nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534911(CHEMBL4454441)
Affinity DataIC50:  9nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534859(CHEMBL4513527)
Affinity DataIC50:  10nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534888(CHEMBL4453133)
Affinity DataIC50:  10nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534914(CHEMBL4458317)
Affinity DataIC50:  12nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534897(CHEMBL4524663)
Affinity DataIC50:  12nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534886(CHEMBL4573137)
Affinity DataIC50:  12nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534861(CHEMBL4526334)
Affinity DataIC50:  15nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534864(CHEMBL4442859)
Affinity DataIC50:  15nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534883(CHEMBL4453296)
Affinity DataIC50:  21nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534901(CHEMBL4591920)
Affinity DataIC50:  22nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534913(CHEMBL4576172)
Affinity DataIC50:  33nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534884(CHEMBL4457643)
Affinity DataIC50:  40nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534896(CHEMBL4518284)
Affinity DataIC50:  41nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534889(CHEMBL4535251)
Affinity DataIC50:  85nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534863(CHEMBL4469642)
Affinity DataIC50:  112nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534882(CHEMBL4544856)
Affinity DataIC50:  120nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534908(CHEMBL4437545)
Affinity DataIC50:  130nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534891(CHEMBL4449211)
Affinity DataIC50:  137nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534877(CHEMBL4464649)
Affinity DataIC50:  200nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534881(CHEMBL4453546)
Affinity DataIC50:  200nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534906(CHEMBL4447542)
Affinity DataIC50:  200nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534878(CHEMBL4466958)
Affinity DataIC50: >200nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534856(CHEMBL4439447)
Affinity DataIC50:  200nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534875(CHEMBL4466826)
Affinity DataIC50:  250nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534880(CHEMBL4543664)
Affinity DataIC50:  300nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534865(CHEMBL4455319)
Affinity DataIC50:  300nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534912(CHEMBL4452080)
Affinity DataIC50:  400nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534900(CHEMBL4451670)
Affinity DataIC50:  400nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534876(CHEMBL4466612)
Affinity DataIC50:  500nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534879(CHEMBL4441620)
Affinity DataIC50:  500nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534905(CHEMBL4583847)
Affinity DataIC50:  800nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of Aberdeen

Curated by ChEMBL
LigandPNGBDBM50534874(CHEMBL4457413)
Affinity DataIC50:  800nMAssay Description:Negative allosteric modulation of human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of CP55940 induced beta arrestin recruitment pr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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