Compile Data Set for Download or QSAR
Report error Found 167 Enz. Inhib. hit(s) with all data for entry = 50047994
LigandChemical structure of BindingDB Monomer ID 50200375BDBM50200375(CHEMBL3902514)
Affinity DataIC50: 10nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200429BDBM50200429(CHEMBL3981511 | US9763922, Example 67)
Affinity DataIC50: 20nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200376BDBM50200376(CHEMBL3896323)
Affinity DataIC50: 20nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200377BDBM50200377(CHEMBL3962542 | US9763922, Example 64)
Affinity DataIC50: 20nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200384BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
Affinity DataIC50: 20nMAssay Description:Displacement of biotinylated ligand from CBP (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200428BDBM50200428(CHEMBL3917504 | US9763922, Example 89)
Affinity DataIC50: 20nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200397BDBM50200397(CHEMBL3973515 | US9763922, Example 79)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200423BDBM50200423(CHEMBL3911524)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200425BDBM50200425(CHEMBL3934488)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200383BDBM50200383(CHEMBL3938408 | US9763922, Example 73)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200430BDBM50200430(CHEMBL3893541 | US9763922, Example 63)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50200384BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200431BDBM50200431(CHEMBL3889679 | US9763922, Example 218)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 50200459BDBM50200459(CHEMBL3920459 | US9763922, Example 71)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200427BDBM50200427(CHEMBL3924330 | US9763922, Example 179)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 188519BDBM188519(SGC-CBP30)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from CBP (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200390BDBM50200390(CHEMBL3892467 | US9763922, Example 70)
Affinity DataIC50: 30nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200424BDBM50200424(CHEMBL3915331)
Affinity DataIC50: 40nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200421BDBM50200421(CHEMBL3985118 | US9763922, Example 173)
Affinity DataIC50: 40nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200378BDBM50200378(CHEMBL3906525)
Affinity DataIC50: 40nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200379BDBM50200379(CHEMBL3962757 | US9763922, Example 201)
Affinity DataIC50: 60nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200384BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
Affinity DataEC50:  69nMAssay Description:Inhibition of CBP/EP300 in human MOLM16 cells assessed as decrease in MYC expression measured after 4 hrs by RT-PCR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200455BDBM50200455(CHEMBL3915504 | US9763922, Example 219)
Affinity DataIC50: 70nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200426BDBM50200426(CHEMBL3980755)
Affinity DataIC50: 70nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200398BDBM50200398(CHEMBL3910675 | US9763922, Example 199)
Affinity DataIC50: 90nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200389BDBM50200389(CHEMBL3936675 | US9763922, Example 195)
Affinity DataIC50: 90nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200381BDBM50200381(CHEMBL3898753)
Affinity DataIC50: 100nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200440BDBM50200440(CHEMBL3907779)
Affinity DataIC50: 110nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200435BDBM50200435(CHEMBL3897524 | US9763922, Example 203)
Affinity DataIC50: 140nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200453BDBM50200453(CHEMBL3926801)
Affinity DataIC50: 140nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200434BDBM50200434(CHEMBL3986361 | US9763922, Example 196)
Affinity DataIC50: 140nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200444BDBM50200444(CHEMBL3900573 | US9763922, Example 217)
Affinity DataIC50: 150nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200438BDBM50200438(CHEMBL3891644)
Affinity DataIC50: 160nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200386BDBM50200386(CHEMBL3909879)
Affinity DataIC50: 180nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Genentech

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 188517BDBM188517(PF-CBP1)
Affinity DataIC50: 190nMAssay Description:Displacement of biotinylated ligand from CBP (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200422BDBM50200422(CHEMBL3963381)
Affinity DataIC50: 190nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200433BDBM50200433(CHEMBL3916599 | US9763922, Example 202)
Affinity DataIC50: 200nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200387BDBM50200387(CHEMBL3972721 | US9763922, Example 198)
Affinity DataIC50: 200nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200391BDBM50200391(CHEMBL3928531 | US9763922, Example 214)
Affinity DataIC50: 220nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200454BDBM50200454(CHEMBL3919629 | US9763922, Example 188)
Affinity DataIC50: 230nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200458BDBM50200458(CHEMBL3935734)
Affinity DataIC50: 250nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200377BDBM50200377(CHEMBL3962542 | US9763922, Example 64)
Affinity DataIC50: 280nMAssay Description:Inhibition of Halo-tagged histone H3.3 binding to CBP/EP300 (unknown origin) expressed in HEK293 cells measured after overnight incubation by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200456BDBM50200456(CHEMBL3899464)
Affinity DataIC50: 300nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200452BDBM50200452(CHEMBL3891576 | US9763922, Example 204)
Affinity DataIC50: 310nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200390BDBM50200390(CHEMBL3892467 | US9763922, Example 70)
Affinity DataIC50: 330nMAssay Description:Inhibition of Halo-tagged histone H3.3 binding to CBP/EP300 (unknown origin) expressed in HEK293 cells measured after overnight incubation by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200443BDBM50200443(CHEMBL3970636)
Affinity DataIC50: 340nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200429BDBM50200429(CHEMBL3981511 | US9763922, Example 67)
Affinity DataIC50: 340nMAssay Description:Inhibition of Halo-tagged histone H3.3 binding to CBP/EP300 (unknown origin) expressed in HEK293 cells measured after overnight incubation by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200439BDBM50200439(CHEMBL3917847)
Affinity DataIC50: 340nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200457BDBM50200457(CHEMBL3943463 | US9763922, Example 220)
Affinity DataIC50: 360nMAssay Description:Displacement of biotinylated ligand from recombinant His-tagged CBP/EP300 (unknown origin) measured after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50200384BDBM50200384(CHEMBL3968533 | US9763922, Example 299)
Affinity DataIC50: 400nMAssay Description:Inhibition of Halo-tagged histone H3.3 binding to CBP/EP300 (unknown origin) expressed in HEK293 cells measured after overnight incubation by lucifer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2018
Entry Details Article
PubMed
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