Compile Data Set for Download or QSAR
maximum 50k data
Found 23 Enz. Inhib. hit(s) with all data for entry = 50049112
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234631(CHEMBL4078686)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234634(CHEMBL4100259)
Affinity DataIC50:  17nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234638(CHEMBL4092511)
Affinity DataIC50:  22nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50069985((S)-4-methyl-2-(3-phenyl-propionylamino)-pentanoic...)
Affinity DataIC50:  25nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234630(CHEMBL4077762)
Affinity DataIC50:  1.36E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234655(CHEMBL4102028)
Affinity DataIC50:  1.97E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234653(CHEMBL4066773)
Affinity DataIC50:  2.71E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234641(CHEMBL4093360)
Affinity DataIC50:  3.57E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234654(CHEMBL4072644)
Affinity DataIC50:  5.84E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234636(CHEMBL4083790)
Affinity DataIC50:  8.83E+3nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234634(CHEMBL4100259)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using (Z)-LLE-bNA as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234635(CHEMBL4073408)
Affinity DataIC50:  1.96E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234659(CHEMBL4062055)
Affinity DataIC50:  2.22E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234639(CHEMBL4064046)
Affinity DataIC50:  2.23E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234636(CHEMBL4083790)
Affinity DataIC50:  2.26E+4nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using (Z)-LLE-bNA as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234638(CHEMBL4092511)
Affinity DataIC50:  2.27E+4nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using (Z)-LLE-bNA as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234642(CHEMBL4094297)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234631(CHEMBL4078686)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of PGPH activity of human 20S proteasome using (Z)-LLE-bNA as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234637(CHEMBL4070680)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234633(CHEMBL4064812)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234632(CHEMBL4096708)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234638(CHEMBL4092511)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of trypsin-like activity of human 20S proteasome using Bz-VGR-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Guangxi Normal University

Curated by ChEMBL
LigandPNGBDBM50234640(CHEMBL4085613)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of chymotrypsin-like activity of human 20S proteasome using Suc-LLVY-AMC as substrate by fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed