Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50006632
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501361BDBM50501361(CHEMBL4097746)
Affinity DataIC50: 8.94E+3nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501368BDBM50501368(CHEMBL4074006)
Affinity DataIC50: 1.07E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 23926BDBM23926(5-[(E)-2-(4-hydroxyphenyl)ethenyl]benzene-1,3-diol...)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501363BDBM50501363(CHEMBL4086825)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501364BDBM50501364(CHEMBL4068105)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501362BDBM50501362(CHEMBL4070599)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50140172BDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501366BDBM50501366(CHEMBL4059796)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501359BDBM50501359(CHEMBL4077009)
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501365BDBM50501365(CHEMBL4095488)
Affinity DataIC50: 2.18E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501367BDBM50501367(CHEMBL4074429)
Affinity DataIC50: 2.34E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed
TargetAmyloid-beta precursor protein(Human)
Zhejiang Chinese Medical University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50501360BDBM50501360(CHEMBL4092433)
Affinity DataIC50: 2.92E+4nMAssay Description:Inhibition of HFIP-pretreated amyloid beta (1 to 42) (unknown origin) self-induced aggregation incubated for 24 hrs under dark condition by thioflavi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2020
Entry Details Article
PubMed