Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50048205
TargetMu-type opioid receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50081529((S)-2-Amino-N-{(R)-1-[({(S)-2-[N'-((S)-2-amino-3-p...)
Affinity DataIC50: 0.740nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetSubstance-P receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50001450(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met NH2 | ...)
Affinity DataIC50: 1.10nMAssay Description:Displacement of [Leu-3,4,5-3H(N)]-Substance P from NK1 receptor in rat brain homogenate measured after 60 mins by microbeta scintillation counting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50208162(CHEMBL3904919)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50208162(CHEMBL3904919)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetSubstance-P receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50: 4.20nMAssay Description:Displacement of [Leu-3,4,5-3H(N)]-Substance P from NK1 receptor in rat brain homogenate measured after 60 mins by microbeta scintillation counting an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50081523((S)-2-Amino-N-((R)-1-{[((S)-1-hydrazinocarbonyl-2-...)
Affinity DataIC50: 4.70nMAssay Description:Displacement of [3H]DAMGO from MOR in Sprague-Dawley rat brain homogenate measured after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50: 13nMAssay Description:Displacement of [3H]DAMGO from MOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50081529((S)-2-Amino-N-{(R)-1-[({(S)-2-[N'-((S)-2-amino-3-p...)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50208161(CHEMBL3932836)
Affinity DataIC50: 74nMAssay Description:Displacement of [3H]DELT2 from DOR in rat brain homogenate measured after 60 mins by microbeta scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
Mossakowski Medical Research Centre Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50081523((S)-2-Amino-N-((R)-1-{[((S)-1-hydrazinocarbonyl-2-...)
Affinity DataIC50: 230nMAssay Description:Displacement of [3H]DELT2 from DOR in Sprague-Dawley rat brain homogenate measured after 180 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2018
Entry Details Article
PubMed