Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50000293
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM185181(N-[2-[4-[[5-(dimethylamino)-1-naphthyl]sulfonyl]pi...)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human TG2 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2019
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50444514(CHEMBL3092843)
Affinity DataIC50: 20nMAssay Description:Inhibition of human TG2 using glycine methyl ester/Abz-APE as substrate after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2019
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50444513(CHEMBL3092841)
Affinity DataIC50: 30nMAssay Description:Inhibition of human TG2 using glycine methyl ester/Abz-APE as substrate after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2019
Entry Details Article
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Daegu-Gyeongbuk Medical Innovation Foundation (Dgmif)

Curated by ChEMBL
LigandPNGBDBM50245478(CHEMBL4081588 | US11472838, Compound Ref. 25)
Affinity DataIC50: 45nMAssay Description:Inhibition of human TG2 using glycine methyl ester/Abz-APE as substrate after 5 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/25/2019
Entry Details Article
PubMed