Compile Data Set for Download or QSAR
Report error Found 111 Enz. Inhib. hit(s) with all data for entry = 50049218
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50318633BDBM50318633(SB-742457 | 3-benzenesulfonyl-8-piperazin-1-ylquin...)
Affinity DataKi:  0.230nMAssay Description:Antagonist activity at 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50019754BDBM50019754(LU-AE58054 | IDALOPIRDINE)
Affinity DataKi:  0.830nMAssay Description:Antagonist activity at 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50044616BDBM50044616(Cerlapirdine | PF-05212365 | SAM-531 | WAY-262531)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at 5-HT6 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236846BDBM50236846(CHEMBL4080401)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236844BDBM50236844(CHEMBL4100484)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236780BDBM50236780(CHEMBL4068232)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236756BDBM50236756(CHEMBL4101284)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236754BDBM50236754(CHEMBL4082473)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236773BDBM50236773(CHEMBL4065437)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236832BDBM50236832(CHEMBL4093699)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236806BDBM50236806(CHEMBL4100411)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236831BDBM50236831(CHEMBL4077537)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236836BDBM50236836(CHEMBL4073586)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236792BDBM50236792(CHEMBL4083289)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236843BDBM50236843(CHEMBL4105377)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236833BDBM50236833(CHEMBL4062687)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236777BDBM50236777(CHEMBL4097459)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236821BDBM50236821(CHEMBL4075502)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236834BDBM50236834(CHEMBL4073450)
Affinity DataKi:  6.90nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236803BDBM50236803(CHEMBL4095054)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236801BDBM50236801(CHEMBL4092681)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236810BDBM50236810(CHEMBL4103281)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236839BDBM50236839(CHEMBL4083893)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236812BDBM50236812(CHEMBL4070284)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236793BDBM50236793(CHEMBL4064478)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236808BDBM50236808(CHEMBL4071816)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236788BDBM50236788(CHEMBL4085949)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236829BDBM50236829(CHEMBL4087957)
Affinity DataKi:  9.60nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236798BDBM50236798(CHEMBL4064995)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236770BDBM50236770(CHEMBL4074058)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236847BDBM50236847(CHEMBL4085003)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236769BDBM50236769(CHEMBL4066125)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236851BDBM50236851(CHEMBL4079859)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236841BDBM50236841(CHEMBL4101418)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236776BDBM50236776(CHEMBL4091721)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236852BDBM50236852(CHEMBL4093110)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236820BDBM50236820(CHEMBL4103877)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236845BDBM50236845(CHEMBL4060415)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236819BDBM50236819(CHEMBL4074732)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236816BDBM50236816(CHEMBL4070850)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236813BDBM50236813(CHEMBL4090177)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236800BDBM50236800(CHEMBL4100818)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236768BDBM50236768(CHEMBL4070785)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236790BDBM50236790(CHEMBL4082319)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236799BDBM50236799(CHEMBL4095670)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236797BDBM50236797(CHEMBL4074234)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236825BDBM50236825(CHEMBL4063362)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236755BDBM50236755(CHEMBL4059662)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236849BDBM50236849(CHEMBL4090168)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Suven Life Sciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50236778BDBM50236778(CHEMBL4068056)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]-LSD from recombinant human 5-HT6 receptor expressed in HEK293 cells after 60 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2019
Entry Details Article
PubMed
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