Compile Data Set for Download or QSAR
Report error Found 50 Enz. Inhib. hit(s) with all data for entry = 50000934
LigandChemical structure of BindingDB Monomer ID 50264847BDBM50264847(CHEMBL4096902)
Affinity DataIC50: 0.180nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256209BDBM50256209(CHEMBL4101768)
Affinity DataIC50: 0.190nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264846BDBM50264846(CHEMBL4066531)
Affinity DataIC50: 0.210nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192809BDBM50192809(CHEMBL3941914)
Affinity DataIC50: 0.220nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256228BDBM50256228(CHEMBL4099293)
Affinity DataIC50: 0.290nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192811BDBM50192811(CHEMBL3971502)
Affinity DataIC50: 0.300nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264858BDBM50264858(CHEMBL4077638)
Affinity DataIC50: 0.310nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264859BDBM50264859(CHEMBL4078117)
Affinity DataIC50: 0.390nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192809BDBM50192809(CHEMBL3941914)
Affinity DataIC50: 0.400nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of hypotonicity-induced activation pretreated for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264845BDBM50264845(CHEMBL4095552)
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256212BDBM50256212(CHEMBL4060956)
Affinity DataIC50: 0.620nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264848BDBM50264848(CHEMBL4062935)
Affinity DataIC50: 0.650nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264857BDBM50264857(CHEMBL4090714)
Affinity DataIC50: 0.710nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of hypotonicity-induced activation pretreated for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264856BDBM50264856(CHEMBL4084992)
Affinity DataIC50: 0.870nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256230BDBM50256230(CHEMBL4083772)
Affinity DataIC50: 0.970nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264855BDBM50264855(CHEMBL4091558)
Affinity DataIC50: 0.990nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264844BDBM50264844(CHEMBL4069724)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of hypotonicity-induced activation pretreated for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256210BDBM50256210(CHEMBL4080527)
Affinity DataIC50: 1.30nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50263440BDBM50263440(CHEMBL4083195)
Affinity DataIC50: 1.40nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of hypotonicity-induced activation pretreated for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256211BDBM50256211(CHEMBL4077429)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50133817BDBM50133817(BCTC | CHEMBL441472 | N-(4-tert-butylphenyl)-4-(3-...)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256229BDBM50256229(CHEMBL4063752)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50263440BDBM50263440(CHEMBL4083195)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264844BDBM50264844(CHEMBL4069724)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256213BDBM50256213(CHEMBL4082835)
Affinity DataIC50: 2.40nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264857BDBM50264857(CHEMBL4090714)
Affinity DataIC50: 2.60nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264868BDBM50264868(CHEMBL4075898)
Affinity DataIC50: 3.70nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50263438BDBM50263438(CHEMBL4077357)
Affinity DataIC50: 3.90nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264860BDBM50264860(CHEMBL4069627)
Affinity DataIC50: 4.20nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256209BDBM50256209(CHEMBL4101768)
Affinity DataIC50: 4.40nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256231BDBM50256231(CHEMBL4077790)
Affinity DataIC50: 6.20nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256208BDBM50256208(CHEMBL4103303)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264850BDBM50264850(CHEMBL4090643)
Affinity DataIC50: 6.80nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256228BDBM50256228(CHEMBL4099293)
Affinity DataIC50: 8.20nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192809BDBM50192809(CHEMBL3941914)
Affinity DataIC50: 8.60nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256212BDBM50256212(CHEMBL4060956)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256208BDBM50256208(CHEMBL4103303)
Affinity DataIC50: 23nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of hypotonicity-induced activation pretreated for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192821BDBM50192821(CHEMBL2133556)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of hypotonicity-induced activation pretreated for 5 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256211BDBM50256211(CHEMBL4077429)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256210BDBM50256210(CHEMBL4080527)
Affinity DataIC50: 39nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256229BDBM50256229(CHEMBL4063752)
Affinity DataIC50: 47nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256230BDBM50256230(CHEMBL4083772)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192821BDBM50192821(CHEMBL2133556)
Affinity DataIC50: 57nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256213BDBM50256213(CHEMBL4082835)
Affinity DataIC50: 62nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264854BDBM50264854(CHEMBL4072343)
Affinity DataIC50: 64nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50264849BDBM50264849(CHEMBL4076956)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at recombinant human TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192821BDBM50192821(CHEMBL2133556)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256231BDBM50256231(CHEMBL4077790)
Affinity DataIC50: 180nMAssay Description:Antagonist activity at recombinant rat TRPV4 expressed in CHOK1 cells assessed as inhibition of 4alphaPDD-induced activation pretreated for 5 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50192809BDBM50192809(CHEMBL3941914)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50256209BDBM50256209(CHEMBL4101768)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/9/2020
Entry Details Article
PubMed