Compile Data Set for Download or QSAR
maximum 50k data
Found 84 Enz. Inhib. hit(s) with all data for entry = 50049287
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50:  64nMAssay Description:Inhibition of human CREBBP by FRET assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238139(CHEMBL4066064)
Affinity DataIC50:  76nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238135(CHEMBL4074125)
Affinity DataIC50:  90nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM188516(BDOIA383)
Affinity DataIC50:  120nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238128(CHEMBL4101368)
Affinity DataIC50:  130nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM188517(PF-CBP1)
Affinity DataIC50:  130nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238153(CHEMBL4066476)
Affinity DataIC50:  130nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238138(CHEMBL4093638)
Affinity DataIC50:  140nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238130(CHEMBL4063290)
Affinity DataIC50:  160nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238149(CHEMBL4074405)
Affinity DataIC50:  170nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238152(CHEMBL4075074)
Affinity DataIC50:  200nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238134(CHEMBL4085966)
Affinity DataIC50:  200nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238260(CHEMBL4094643)
Affinity DataIC50:  210nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238146(CHEMBL4103593)
Affinity DataIC50:  210nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238262(CHEMBL4094017)
Affinity DataIC50:  240nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238255(CHEMBL3753333)
Affinity DataIC50:  240nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238259(CHEMBL4096429)
Affinity DataIC50:  240nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238151(CHEMBL4063726)
Affinity DataIC50:  260nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238136(CHEMBL4065507)
Affinity DataIC50:  300nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238142(CHEMBL4078019)
Affinity DataIC50:  310nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238258(CHEMBL4075476)
Affinity DataIC50:  310nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238263(CHEMBL4064489)
Affinity DataIC50:  330nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238146(CHEMBL4103593)
Affinity DataIC50:  350nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238261(CHEMBL4074676)
Affinity DataIC50:  360nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238131(CHEMBL4077279)
Affinity DataIC50:  400nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238254(CHEMBL4104158)
Affinity DataIC50:  400nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238140(CHEMBL4085900)
Affinity DataIC50:  450nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238256(CHEMBL4078384)
Affinity DataIC50:  470nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238139(CHEMBL4066064)
Affinity DataIC50:  490nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238148(CHEMBL4078551)
Affinity DataIC50:  500nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238145(CHEMBL4068497)
Affinity DataIC50:  500nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM188517(PF-CBP1)
Affinity DataIC50:  620nMAssay Description:Displacement of [3H]prazosin from recombinant human adrenergic A1a receptor after 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238133(CHEMBL4071814)
Affinity DataIC50:  650nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238150(CHEMBL4085329)
Affinity DataIC50:  690nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238264(CHEMBL4068021)
Affinity DataIC50:  740nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238132(CHEMBL4092184)
Affinity DataIC50:  780nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238253(CHEMBL4086250)
Affinity DataIC50:  920nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238257(CHEMBL4095141)
Affinity DataIC50:  980nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238141(CHEMBL4103824)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238134(CHEMBL4085966)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238147(CHEMBL4076179)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238133(CHEMBL4071814)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238128(CHEMBL4101368)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238140(CHEMBL4085900)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM188516(BDOIA383)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238143(CHEMBL4096066)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238129(CHEMBL4084942)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238263(CHEMBL4064489)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238135(CHEMBL4074125)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238145(CHEMBL4068497)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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