Compile Data Set for Download or QSAR
Report error Found 207 Enz. Inhib. hit(s) with all data for entry = 50000104
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240674(CHEMBL4097965)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240613(CHEMBL4074974)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240638(CHEMBL4066368)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240651(CHEMBL3276119)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240632(CHEMBL4070222)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240633(CHEMBL4093631)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240610(CHEMBL4101658)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50044752(CHEMBL3353956)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataEC50:  0.00800nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240636(CHEMBL4104080)
Affinity DataEC50:  0.00800nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50044676(CHEMBL439044)
Affinity DataEC50:  0.00900nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240634(CHEMBL4074335)
Affinity DataEC50:  0.00900nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240630(CHEMBL4102192)
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240644(CHEMBL3277916)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240607(CHEMBL4093931)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240672(CHEMBL4095930)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240629(CHEMBL4084223)
Affinity DataEC50:  0.0140nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240663(CHEMBL4078856)
Affinity DataEC50:  0.0150nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240673(CHEMBL4096848)
Affinity DataEC50:  0.0210nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240675(CHEMBL4101771)
Affinity DataEC50:  0.0270nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240631(CHEMBL4065273)
Affinity DataEC50:  0.0270nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240628(CHEMBL4094454)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240604(CHEMBL4092971)
Affinity DataEC50:  0.0310nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240628(CHEMBL4094454)
Affinity DataEC50:  0.0340nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240646(CHEMBL4080341)
Affinity DataEC50:  0.0420nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240647(CHEMBL4084795)
Affinity DataEC50:  0.0540nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240649(CHEMBL4063150)
Affinity DataEC50:  0.0560nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240661(CHEMBL3277915)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240665(CHEMBL4101586)
Affinity DataEC50:  0.0720nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240640(CHEMBL4065416)
Affinity DataEC50:  0.0820nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240645(CHEMBL4066923)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240595(CHEMBL4070577)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240666(CHEMBL4093088)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240628(CHEMBL4094454)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human V1a receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240637(CHEMBL4096331)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50147625(CHEBI:16136 | SULFUR, PRECIPITATED | BDBM50498447)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240635(CHEMBL4075102)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240673(CHEMBL4096848)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240639(CHEMBL4083700)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240600(CHEMBL4092407)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240667(CHEMBL4100627)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240627(CHEMBL4073891)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240603(CHEMBL4072207)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240641(CHEMBL4092242)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240595(CHEMBL4070577)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240663(CHEMBL4078856)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetOxytocin receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240626(CHEMBL4099102)
Affinity DataEC50:  0.530nMAssay Description:Agonist activity at human OTR expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240675(CHEMBL4101771)
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240631(CHEMBL4065273)
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50240649(CHEMBL4063150)
Affinity DataEC50:  0.650nMAssay Description:Agonist activity at human V1b receptor expressed in CHO cells assessed as calcium mobilization measured after 30 mins by Fluo-4-AM dye based FLIPR as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2019
Entry Details Article
PubMed
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