Compile Data Set for Download or QSAR
maximum 50k data
Found 36 Enz. Inhib. hit(s) with all data for entry = 50001129
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269809(CHEMBL4077195)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of human LRRK2 using RLGRDKYKTLRQIRQ as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269801(CHEMBL4100294)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269824(CHEMBL4098650)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269800(CHEMBL4068065)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269816(CHEMBL4072195)
Affinity DataIC50:  10nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269810(CHEMBL4101126)
Affinity DataIC50:  10nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM482159(BDBM50401284 | GSK2578215A)
Affinity DataIC50:  10nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269823(CHEMBL4071631)
Affinity DataIC50:  10nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269789(CHEMBL4084470)
Affinity DataIC50:  13nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269807(CHEMBL4063006)
Affinity DataIC50:  13nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269819(CHEMBL4082330)
Affinity DataIC50:  13nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269797(CHEMBL4062430)
Affinity DataIC50:  16nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269814(CHEMBL4066777)
Affinity DataIC50:  16nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269818(CHEMBL4067228)
Affinity DataIC50:  16nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269809(CHEMBL4077195)
Affinity DataIC50:  20nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269790(CHEMBL4073840)
Affinity DataIC50:  20nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269803(CHEMBL4065244)
Affinity DataIC50:  20nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269826(CHEMBL4083585)
Affinity DataIC50:  25nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269792(CHEMBL4094423)
Affinity DataIC50:  40nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269817(CHEMBL4089737)
Affinity DataIC50:  40nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269802(CHEMBL4068792)
Affinity DataIC50:  40nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269804(CHEMBL4086683)
Affinity DataIC50:  50nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269788(CHEMBL4103192)
Affinity DataIC50:  63nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269795(CHEMBL4059881)
Affinity DataIC50:  63nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269799(CHEMBL4088336)
Affinity DataIC50:  100nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269796(CHEMBL4105171)
Affinity DataIC50:  126nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSRSF protein kinase 3(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269809(CHEMBL4077195)
Affinity DataIC50:  158nMAssay Description:Inhibition of human MSSK1 GRSRSRSRSR as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269813(CHEMBL4070845)
Affinity DataIC50:  200nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269825(CHEMBL4076463)
Affinity DataIC50:  251nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269811(CHEMBL4083136)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269805(CHEMBL4090116)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269793(CHEMBL4097465)
Affinity DataIC50:  2.51E+3nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269798(CHEMBL4087313)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269806(CHEMBL4078829)
Affinity DataIC50: <2.51E+4nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269794(CHEMBL4079429)
Affinity DataIC50: <2.51E+4nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu

Curated by ChEMBL
LigandPNGBDBM50269791(CHEMBL4075367)
Affinity DataIC50: <2.51E+4nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed