TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of human LRRK2 using RLGRDKYKTLRQIRQ as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 7.90nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 126nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of human MSSK1 GRSRSRSRSR as substrate in presence of [gamma-33P]-ATPMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 2.51E+3nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: <2.51E+4nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: <2.51E+4nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetLeucine-rich repeat serine/threonine-protein kinase 2(Homo sapiens (Human))
Neurodegeneration Dpu
Curated by ChEMBL
Neurodegeneration Dpu
Curated by ChEMBL
Affinity DataIC50: <2.51E+4nMAssay Description:Inhibition of LRRK2 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair