TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 102nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 112nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 129nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 176nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 221nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 228nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 259nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 267nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 287nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 287nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 351nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 438nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 445nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 565nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 704nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 733nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 766nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 2.36E+3nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 3.23E+3nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 5.91E+3nMAssay Description:Inhibition of ABCB1 in human A2780adr cells assessed as reduction in calcein AM levels preincubated for 30 mins followed by calcein AM addition measu...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 6.91E+3nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 7.67E+3nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 8.34E+3nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 8.55E+3nMAssay Description:Inhibition of ABCB1 in human A2780adr cells assessed as reduction in calcein AM levels preincubated for 30 mins followed by calcein AM addition measu...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of ABCB1 in human A2780adr cells assessed as reduction in calcein AM levels preincubated for 30 mins followed by calcein AM addition measu...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 1.53E+4nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 1.58E+4nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 1.85E+4nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 2.12E+4nMAssay Description:Inhibition of ABCB1 in human A2780adr cells assessed as reduction in calcein AM levels preincubated for 30 mins followed by calcein AM addition measu...More data for this Ligand-Target Pair
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Rheinische Friedrich-Wilhelms-Universit£T Bonn
Curated by ChEMBL
Affinity DataIC50: 3.98E+4nMAssay Description:Inhibition of C-terminal GFP-fused human ABCG2 expressed in MDCK2 cells preincubated for 30 mins followed by Hoechst 33342 addition and measured ever...More data for this Ligand-Target Pair