Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50001697
TargetC-C chemokine receptor type 5(Mouse)
Nirma University

Curated by ChEMBL
LigandPNGBDBM50306033(Cenicriviroc | TAK-652 | TBR-652)
Affinity DataIC50: 0.25nMAssay Description:Displacement of [125I]-RANTES from CCR5 in mouse NIH/3T3 cells after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2020
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Mouse)
Nirma University

Curated by ChEMBL
LigandPNGBDBM50336345(APLAVIROC | CHEMBL1668019 | 4-(4-(((R)-1-butyl-3-(...)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I]-RANTES from CCR5 in mouse NIH/3T3 cells after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2020
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Mouse)
Nirma University

Curated by ChEMBL
LigandPNGBDBM50145685((4,6-Dimethyl-pyrimidin-5-yl)-(4-{(S)-4-[(R)-2-met...)
Affinity DataIC50: 0.910nMAssay Description:Displacement of [125I]-RANTES from CCR5 in mouse NIH/3T3 cells after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2020
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Mouse)
Nirma University

Curated by ChEMBL
LigandPNGBDBM50321682(nifeviroc | CHEMBL1172035)
Affinity DataIC50: 2.90nMAssay Description:Displacement of [125I]-RANTES from CCR5 in mouse NIH/3T3 cells after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2020
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Mouse)
Nirma University

Curated by ChEMBL
LigandPNGBDBM50334986(4,4-Difluoro-cyclohexanecarboxylic acid {(S)-3-[(1...)
Affinity DataIC50: 5.20nMAssay Description:Displacement of [125I]-RANTES from CCR5 in mouse NIH/3T3 cells after 1 hrMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2020
Entry Details Article
PubMed
TargetC-C chemokine receptor type 5(Human)
Nirma University

Curated by ChEMBL
LigandPNGBDBM50306034(CHEMBL4160473)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at CCR5 (unknown origin) by HTS assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2020
Entry Details Article
PubMed