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Found 4 Enz. Inhib. hit(s) with all data for entry = 50006764
TargetProteinase-activated receptor 2(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50274114(CHEMBL4128763)
Affinity DataIC50: <2.5nMAssay Description:Antagonist activity at human PAR2More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 2(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50503155(CHEMBL4519152)
Affinity DataIC50:  170nMAssay Description:Negative allosteric modulation of CCR2 (unknown origin)More data for this Ligand-Target Pair
TargetProteinase-activated receptor 4(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50274114(CHEMBL4128763)
Affinity DataIC50:  380nMAssay Description:Antagonist activity at human PAR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50274114(CHEMBL4128763)
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at human PAR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed