TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 43nMAssay Description:Inverse agonist activity at LXRbeta (unknown origin) expressed in HEK293 cells 24 hrs by Dual-Glo luciferase assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 214nMAssay Description:Inverse agonist activity at LXRalpha (unknown origin) expressed in HEK293 cells 24 hrs by Dual-Glo luciferase assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.50E+3nMAssay Description:Antagonist activity at human LXRalpha expressed in HEK293T cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Agonist activity at human LXRalpha-LBD (182 to 447 amino acids) expressed in HEK293T cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataEC50: 230nMAssay Description:Agonist activity at human LXRalpha expressed in HEK293 cells after 24 hrs by One-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataEC50: 530nMAssay Description:Agonist activity at human LXRbeta-LBD (196 to 461 amino acids) expressed in HEK293T cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataEC50: 108nMAssay Description:Agonist activity at human full length LXRbeta expressed in African green monkey CV-1 cells co-expressing human pCMX/RXRalpha after 20 hrs by lucifera...More data for this Ligand-Target Pair
TargetOxysterols receptor LXR-beta(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataEC50: 720nMAssay Description:Agonist activity at GAL4-tagged human LXRbeta LBD expressed in HEK293T cells after 12 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Saint Louis University School Of Medicine
Curated by ChEMBL
Saint Louis University School Of Medicine
Curated by ChEMBL
Affinity DataEC50: 422nMAssay Description:Agonist activity at human LXRalpha expressed in HEK293 cells after 24 hrs by One-Glo luciferase reporter gene assayMore data for this Ligand-Target Pair