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Found 9 Enz. Inhib. hit(s) with all data for entry = 50002849
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)
Affinity DataIC50:  262nMAssay Description:Inhibition of MNK2 (unknown origin) using S3 as substrate measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50463694(CHEMBL4248798)
Affinity DataIC50:  273nMAssay Description:Inhibition of MNK2 (unknown origin) using S3 as substrate measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50463696(CHEMBL4247747)
Affinity DataIC50:  749nMAssay Description:Inhibition of MNK2 (unknown origin) using S3 as substrate measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50130693(CGP-57380 | CHEMBL1240885)
Affinity DataIC50:  850nMAssay Description:Inhibition of MNK1 (unknown origin) using S3 as substrate measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50463695(CHEMBL4237434)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of MNK2 (unknown origin) using S3 as substrate measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50463697(CHEMBL4238675)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of MNK2 (unknown origin) using S3 as substrate measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50130693(CGP-57380 | CHEMBL1240885)
Affinity DataIC50:  1.53E+3nMAssay Description:Inhibition of MNK2 (unknown origin) using S3 as substrate measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50130693(CGP-57380 | CHEMBL1240885)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of MNK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Homo sapiens (Human))
Shenyang Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50463693(CHEMBL4249658)
Affinity DataIC50:  3.55E+3nMAssay Description:Inhibition of MNK2 (unknown origin) using S3 as substrate measured after 60 mins by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed