Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50003100
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466974(CHEMBL4285413)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466983(CHEMBL4277337)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466970(CHEMBL4278696)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466984(CHEMBL4284597)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466976(CHEMBL4281986)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466973(CHEMBL4289069)
Affinity DataKi:  52nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466982(CHEMBL4277464)
Affinity DataKi:  59nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466972(CHEMBL4292596)
Affinity DataKi:  67nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466979(CHEMBL4285685)
Affinity DataKi:  76nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466980(CHEMBL4294491)
Affinity DataKi:  77nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466977(CHEMBL4287975)
Affinity DataKi:  95nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466978(CHEMBL4284278)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466975(CHEMBL4277744)
Affinity DataKi:  143nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466971(CHEMBL4281185)
Affinity DataKi:  187nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466981(CHEMBL4283915)
Affinity DataKi:  228nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466983(CHEMBL4277337)
Affinity DataKi:  285nMAssay Description:Displacement of [3H]-(+)-pentazocine from sigma1 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466978(CHEMBL4284278)
Affinity DataKi:  422nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466970(CHEMBL4278696)
Affinity DataKi:  825nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466980(CHEMBL4294491)
Affinity DataKi:  987nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466974(CHEMBL4285413)
Affinity DataKi:  1.12E+3nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466972(CHEMBL4292596)
Affinity DataKi:  1.26E+3nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466984(CHEMBL4284597)
Affinity DataKi:  1.38E+3nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466979(CHEMBL4285685)
Affinity DataKi:  1.84E+3nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466973(CHEMBL4289069)
Affinity DataKi:  2.34E+3nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466977(CHEMBL4287975)
Affinity DataKi:  2.43E+3nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466975(CHEMBL4277744)
Affinity DataKi:  2.58E+3nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSigma intracellular receptor 2(Rattus norvegicus (Rat))
University Of Trieste

Curated by ChEMBL
LigandPNGBDBM50466971(CHEMBL4281185)
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [3H]-DTG from sigma2 receptor in rat liver membranes after 120 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed