Compile Data Set for Download or QSAR
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Found 60 Enz. Inhib. hit(s) with all data for entry = 50002489
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459208(CHEMBL4214342)
Affinity DataIC50:  1nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459215(CHEMBL4202685)
Affinity DataIC50:  2nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459203(CHEMBL4207036)
Affinity DataIC50:  2nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459219(CHEMBL4207100)
Affinity DataIC50:  5nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459216(CHEMBL4213673)
Affinity DataIC50:  5nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459203(CHEMBL4207036)
Affinity DataIC50:  6nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459201(CHEMBL4217421)
Affinity DataIC50:  6nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459211(CHEMBL4214863)
Affinity DataIC50:  7nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459209(CHEMBL4209948)
Affinity DataIC50:  8nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459212(CHEMBL4207753)
Affinity DataIC50:  8nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50323777(CHEMBL1214141 | N-(4-Methyl-3-(1-methyl-7-(6-methy...)
Affinity DataIC50:  8nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459208(CHEMBL4214342)
Affinity DataIC50:  8nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459216(CHEMBL4213673)
Affinity DataIC50:  9nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459218(CHEMBL4211976)
Affinity DataIC50:  10nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459198(CHEMBL4212150)
Affinity DataIC50:  10nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459207(CHEMBL4212663)
Affinity DataIC50:  11nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459215(CHEMBL4202685)
Affinity DataIC50:  13nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459200(CHEMBL4213019)
Affinity DataIC50:  14nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459199(CHEMBL4215916)
Affinity DataIC50:  15nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459221(CHEMBL4216786)
Affinity DataIC50:  16nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459207(CHEMBL4212663)
Affinity DataIC50:  17nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50242740(CHEMBL459850 | N-(3-(7-Amino-1-methyl-2-oxo-1,2-di...)
Affinity DataIC50:  18nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459201(CHEMBL4217421)
Affinity DataIC50:  20nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459213(CHEMBL4212809)
Affinity DataIC50:  20nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459209(CHEMBL4209948)
Affinity DataIC50:  20nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459200(CHEMBL4213019)
Affinity DataIC50:  21nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459197(CHEMBL4209082)
Affinity DataIC50:  21nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459214(CHEMBL4215989)
Affinity DataIC50:  21nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459220(CHEMBL4203337)
Affinity DataIC50:  23nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459198(CHEMBL4212150)
Affinity DataIC50:  24nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459212(CHEMBL4207753)
Affinity DataIC50:  25nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50323777(CHEMBL1214141 | N-(4-Methyl-3-(1-methyl-7-(6-methy...)
Affinity DataIC50:  25nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459221(CHEMBL4216786)
Affinity DataIC50:  25nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459217(CHEMBL4218831)
Affinity DataIC50:  26nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459219(CHEMBL4207100)
Affinity DataIC50:  26nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459202(CHEMBL4211880)
Affinity DataIC50:  27nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50242740(CHEMBL459850 | N-(3-(7-Amino-1-methyl-2-oxo-1,2-di...)
Affinity DataIC50:  28nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459211(CHEMBL4214863)
Affinity DataIC50:  28nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459218(CHEMBL4211976)
Affinity DataIC50:  28nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459214(CHEMBL4215989)
Affinity DataIC50:  33nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459220(CHEMBL4203337)
Affinity DataIC50:  34nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459205(CHEMBL4210482)
Affinity DataIC50:  35nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459222(CHEMBL4213945)
Affinity DataIC50:  36nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50323778(CHEMBL1214142 | N-(4-Methyl-3-(1-methyl-2-oxo-7-(p...)
Affinity DataIC50:  37nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459213(CHEMBL4212809)
Affinity DataIC50:  39nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459206(CHEMBL4205942)
Affinity DataIC50:  40nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetActivated CDC42 kinase 1(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459204(CHEMBL4206139)
Affinity DataIC50:  40nMAssay Description:Inhibition of ACK1 (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459205(CHEMBL4210482)
Affinity DataIC50:  42nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50459217(CHEMBL4218831)
Affinity DataIC50:  45nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Homo sapiens (Human))
Korea University

Curated by ChEMBL
LigandPNGBDBM50323778(CHEMBL1214142 | N-(4-Methyl-3-(1-methyl-2-oxo-7-(p...)
Affinity DataIC50:  47nMAssay Description:Inhibition of GCK (unknown origin) by radiometric biochemical kinase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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