Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50003038
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466079(CHEMBL4286124)
Affinity DataKi:  2.60nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50264998(CHEMBL4103458)
Affinity DataKi:  4.90nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50264998(CHEMBL4103458)
Affinity DataKi:  9.80nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466071(CHEMBL4293336)
Affinity DataKi:  13nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466078(CHEMBL4278214)
Affinity DataKi:  14nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466074(CHEMBL4277812)
Affinity DataKi:  17nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466079(CHEMBL4286124)
Affinity DataKi:  22nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50446936(CHEMBL2179834)
Affinity DataKi:  24nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466076(CHEMBL4285511)
Affinity DataKi:  32nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466071(CHEMBL4293336)
Affinity DataKi:  38nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466074(CHEMBL4277812)
Affinity DataKi:  41nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466077(CHEMBL4289555)
Affinity DataKi:  53nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466076(CHEMBL4285511)
Affinity DataKi:  60nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466078(CHEMBL4278214)
Affinity DataKi:  60nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466075(CHEMBL4288467)
Affinity DataKi:  190nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466073(CHEMBL4285107)
Affinity DataKi:  240nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466077(CHEMBL4289555)
Affinity DataKi:  240nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466075(CHEMBL4288467)
Affinity DataKi:  250nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466070(CHEMBL4292938)
Affinity DataKi:  500nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466073(CHEMBL4285107)
Affinity DataKi:  600nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466070(CHEMBL4292938)
Affinity DataKi:  614nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466072(CHEMBL4281675)
Affinity DataKi:  700nMAssay Description:Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50446936(CHEMBL2179834)
Affinity DataKi:  760nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50466072(CHEMBL4281675)
Affinity DataKi:  825nMAssay Description:Inhibition of recombinant human furin using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed