TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 189nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 189nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 212nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 212nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 348nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 348nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 475nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 475nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 488nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 488nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 919nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 919nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 2.12E+3nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 3.69E+3nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 3.69E+3nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 7.41E+3nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 7.41E+3nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 8.72E+4nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
University Of Sharjah
Curated by ChEMBL
University Of Sharjah
Curated by ChEMBL
Affinity DataIC50: 8.72E+4nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate measured after 40 mins in presence of [gamma33P-ATP] by scintillation c...More data for this Ligand-Target Pair