Affinity DataKi: <0.0100nMAssay Description:Inhibition of BCL-2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Inhibition of BCL-XL (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 245nMAssay Description:Inhibition of BCL-W (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40E+3nMAssay Description:Inhibition of BCL-XL (unknown origin) incubated for 15 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Taros Chemicals
Curated by ChEMBL
Taros Chemicals
Curated by ChEMBL
Affinity DataIC50: 12nMAssay Description:Inhibition of CIAP1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: <40nMAssay Description:Inhibition of XIAP (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of BRD4 bromodomain-1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKd: 8.60E+3nMAssay Description:Binding affinity to HSP90 (unknown origin) by WaterLOGSY NMR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 6.00E+6nMAssay Description:Binding affinity to BCL-XL (unknown origin) by 15N HSQC NMR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Inhibition of BCL-2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataKd: 3.00E+5nMAssay Description:Binding affinity to BCL-XL (unknown origin) by 15N HSQC NMR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 250nMAssay Description:Binding affinity to HSP90 (unknown origin) by WaterLOGSY NMR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 4.30E+6nMAssay Description:Binding affinity to BCL-XL (unknown origin) by 15N HSQC NMR analysisMore data for this Ligand-Target Pair