Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50007741
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM242374(US10047093, 8-31 | US9416132, 8-31 | US10392392, E...)
Affinity DataKi:  5nMAssay Description:Inhibition of PIM1 (unknown origin) up to 120 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512177(CHEMBL4451418)
Affinity DataKi:  7.70nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length Pim-1 expressed in Escherichia coli cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50364776(CHEMBL1952329 | CHEMBL1952141)
Affinity DataKi:  12nMAssay Description:Inhibition of PIM1 (unknown origin) up to 120 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512180(CHEMBL4580240)
Affinity DataIC50: 60nMAssay Description:Inhibition of human PIM1 by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512176(CHEMBL4551767)
Affinity DataIC50: 80nMAssay Description:Inhibition of human PIM1 by ELISAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512179(CHEMBL4469896)
Affinity DataIC50: 111nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512175(CHEMBL4517325)
Affinity DataIC50: 150nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512174(CHEMBL4471511)
Affinity DataIC50: 150nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase pim-1(Human)
Nri Institute of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50512178(CHEMBL4591510)
Affinity DataIC50: 434nMAssay Description:Inhibition of PIM1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/20/2021
Entry Details Article
PubMed