Compile Data Set for Download or QSAR
maximum 50k data
Found 40 Enz. Inhib. hit(s) with all data for entry = 50007493
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataIC50:  3.40nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424074(CHEMBL2314747)
Affinity DataIC50:  40nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509944(CHEMBL4438471)
Affinity DataIC50:  76nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509945(CHEMBL4582377)
Affinity DataIC50:  190nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509944(CHEMBL4438471)
Affinity DataIC50:  390nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424076(CHEMBL2314745)
Affinity DataIC50:  410nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424071(CHEMBL2314734)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424077((-)-Tetrahydropalmatine | L-Tetrahydropalmatine | ...)
Affinity DataIC50:  450nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509946(CHEMBL4476383)
Affinity DataIC50:  500nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424074(CHEMBL2314747)
Affinity DataIC50:  630nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509948(CHEMBL4521450)
Affinity DataIC50:  670nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509945(CHEMBL4582377)
Affinity DataIC50:  1.03E+3nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424071(CHEMBL2314734)
Affinity DataIC50:  1.08E+3nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509941(CHEMBL4544045)
Affinity DataIC50:  1.08E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509946(CHEMBL4476383)
Affinity DataIC50:  1.42E+3nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509940(CHEMBL4561303)
Affinity DataIC50:  1.53E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424077((-)-Tetrahydropalmatine | L-Tetrahydropalmatine | ...)
Affinity DataIC50:  1.63E+3nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM82247(8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-b...)
Affinity DataIC50:  2.05E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509948(CHEMBL4521450)
Affinity DataIC50:  2.59E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424076(CHEMBL2314745)
Affinity DataIC50:  3.11E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509943(CHEMBL4528264)
Affinity DataIC50:  3.58E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509939(CHEMBL4551037)
Affinity DataIC50:  4.94E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509947(CHEMBL4585730)
Affinity DataIC50:  6.36E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509940(CHEMBL4561303)
Affinity DataIC50:  6.51E+3nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509941(CHEMBL4544045)
Affinity DataIC50:  7.42E+3nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424065(CHEMBL2314740)
Affinity DataIC50:  7.96E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509938(CHEMBL4453330)
Affinity DataIC50:  8.81E+3nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509942(CHEMBL4435291)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424063(CHEMBL2314742)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424064(CHEMBL2314741)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424065(CHEMBL2314740)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424063(CHEMBL2314742)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of dopamine-induced calcium flux preincubated for...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509943(CHEMBL4528264)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50424064(CHEMBL2314741)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509942(CHEMBL4435291)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509939(CHEMBL4551037)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509938(CHEMBL4453330)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM50509947(CHEMBL4585730)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as inhibition of SKF38393-induced cAMP accumulation measured af...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM442801(WAY-308264)
Affinity DataEC50:  666nMAssay Description:Agonist activity at D1 receptor (unknown origin) expressed in CHOK1 cells assessed as increase in cAMP accumulation measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Huzhou University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataEC50:  0.990nMAssay Description:Agonist activity at D2 receptor (unknown origin) expressed in CHOK1 cells assessed as increase in calcium flux incubated for 60 mins at 37 degC follo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank