Affinity DataIC50: 0.960nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
Affinity DataIC50: 177nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
Affinity DataIC50: 755nMAssay Description:Inhibition of human MetAP2More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of [3H]Mesulergine from recombinant human 5-HT2C receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 4.40E+3nMAssay Description:Competitive inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of [3H]Mesulergine from recombinant human 5-HT2C receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of [3H]LSD from human 5-HT6 receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of [3H]LSD from human 5-HT7 receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Competitive inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Northwest University
Curated by ChEMBL
Northwest University
Curated by ChEMBL
Affinity DataIC50: 6.70E+3nMAssay Description:Displacement of [3H]Imipramine from human 5-HT transporter expressed in HEK-293 cell membranes after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 6.80E+3nMAssay Description:Displacement of [3H]Ketanserin from recombinant human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from recombinant human 5-HT1A receptor expressed in CHO-K1 cell membranes after 60 mins by microbeta counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80E+3nMAssay Description:Displacement of [3H]Mesulergine from recombinant human 5-HT2C receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10E+3nMAssay Description:Competitive inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 9.40E+3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor (unknown origin) expressed in CHO-K1 cell membranes after 60 mins by microbeta counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5-HT6 receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Northwest University
Curated by ChEMBL
Northwest University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]Imipramine from human 5-HT transporter expressed in HEK-293 cell membranes after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5-HT7 receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from recombinant human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Northwest University
Curated by ChEMBL
Northwest University
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]Imipramine from human 5-HT transporter expressed in HEK-293 cell membranes after 30 minsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5-HT7 receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]Ketanserin from recombinant human 5-HT2A receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]LSD from human 5-HT6 receptor expressed in CHO-K1 cell membranes after 60 minsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+4nMAssay Description:Competitive inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.72E+4nMAssay Description:Competitive inhibition of soluble epoxide hydrolase (unknown origin)More data for this Ligand-Target Pair