Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50008845
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50400272BDBM50400272(CHEMBL2180727)
Affinity DataIC50: 82nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522839BDBM50522839(DNDI1417825 | CHEMBL2095003)
Affinity DataIC50: 410nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522839BDBM50522839(DNDI1417825 | CHEMBL2095003)
Affinity DataKd:  720nMAssay Description:Binding affinity to N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in BL21 cells assessed as equilibrium dissociation constant ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522834BDBM50522834(CHEMBL4570376)
Affinity DataIC50: 800nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522839BDBM50522839(DNDI1417825 | CHEMBL2095003)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522838BDBM50522838(CHEMBL4451545)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522846BDBM50522846(CHEMBL4574726)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522839BDBM50522839(DNDI1417825 | CHEMBL2095003)
Affinity DataKd:  3.80E+3nMAssay Description:Binding affinity to N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in BL21 cells assessed as equilibrium dissociation constant ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522834BDBM50522834(CHEMBL4570376)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522838BDBM50522838(CHEMBL4451545)
Affinity DataIC50: 4.76E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522849BDBM50522849(CHEMBL4556155)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522846BDBM50522846(CHEMBL4574726)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522849BDBM50522849(CHEMBL4556155)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522838BDBM50522838(CHEMBL4451545)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522842BDBM50522842(CHEMBL4456155)
Affinity DataIC50: 8.50E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522842BDBM50522842(CHEMBL4456155)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522847BDBM50522847(CHEMBL4450318)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522849BDBM50522849(CHEMBL4556155)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522847BDBM50522847(CHEMBL4450318)
Affinity DataIC50: 1.27E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522844BDBM50522844(CHEMBL4464973)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522834BDBM50522834(CHEMBL4570376)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522844BDBM50522844(CHEMBL4464973)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522839BDBM50522839(DNDI1417825 | CHEMBL2095003)
Affinity DataIC50: 4.37E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522836BDBM50522836(CHEMBL4539487)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522835BDBM50522835(CHEMBL4584017)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522837BDBM50522837(CHEMBL4524603)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522847BDBM50522847(CHEMBL4450318)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522848BDBM50522848(CHEMBL4455478)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522848BDBM50522848(CHEMBL4455478)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522843BDBM50522843(CHEMBL4446512)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522845BDBM50522845(CHEMBL4448094)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522835BDBM50522835(CHEMBL4584017)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522848BDBM50522848(CHEMBL4455478)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522846BDBM50522846(CHEMBL4574726)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522836BDBM50522836(CHEMBL4539487)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522841BDBM50522841(CHEMBL4558918)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522842BDBM50522842(CHEMBL4456155)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522839BDBM50522839(DNDI1417825 | CHEMBL2095003)
Affinity DataKd: >5.00E+4nMAssay Description:Binding affinity to N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in BL21 cells assessed as equilibrium dissociation constant by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522840BDBM50522840(CHEMBL4537226)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522837BDBM50522837(CHEMBL4524603)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522835BDBM50522835(CHEMBL4584017)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522836BDBM50522836(CHEMBL4539487)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522840BDBM50522840(CHEMBL4537226)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522841BDBM50522841(CHEMBL4558918)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged wild type IDH1 (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in presenc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522837BDBM50522837(CHEMBL4524603)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522845BDBM50522845(CHEMBL4448094)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522843BDBM50522843(CHEMBL4446512)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522840BDBM50522840(CHEMBL4537226)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522841BDBM50522841(CHEMBL4558918)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132C mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetIsocitrate dehydrogenase [NADP] cytoplasmic(Human)
Huazhong Agricultural University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50522845BDBM50522845(CHEMBL4448094)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of N-terminal 6-His-tagged IDH1 R132H mutant (unknown origin) expressed in Escherichia coli BL21 cells using alpha-KG as substrate in pres...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
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