Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50011762
TargetProtein disulfide-isomerase A3(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase A6(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50:  5.70E+3nMAssay Description:Inhibition of PDIA6 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase A6(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of PDIA6 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThioredoxin domain-containing protein 5(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50:  1.21E+4nMAssay Description:Inhibition of TXNDC5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase A6(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50:  1.63E+4nMAssay Description:Inhibition of PDIA6 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase A3(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50:  1.65E+4nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase A3(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of PDIA3 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase A4(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550835(CHEMBL4751979)
Affinity DataIC50:  3.31E+4nMAssay Description:Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase A4(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50:  6.16E+4nMAssay Description:Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThioredoxin domain-containing protein 5(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TXNDC5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThioredoxin domain-containing protein 5(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550836(CHEMBL4751241)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of TXNDC5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein disulfide-isomerase A4(Homo sapiens)
Medical University Of South Carolina

Curated by ChEMBL
LigandPNGBDBM50550837(CHEMBL4762045)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of PDIA4 (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 1 hr and measured by insulin reduction assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed