Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50011093
TargetGlutamate carboxypeptidase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50544832(CHEMBL4636677)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]MIP-1095 from PSMA in human PC3-PIP cells after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50544834(CHEMBL4636963)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MIP-1095 from PSMA in human PC3-PIP cells after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50544835(CHEMBL4649277)
Affinity DataIC50: 2.60nMAssay Description:Displacement of [125I]MIP-1095 from PSMA in human PC3-PIP cells after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50265783((S)-2-(3-((S)-1-Carboxy-5-(3-(4-iodophenyl)ureido)...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]MIP-1095 from PSMA in human PC3-PIP cells after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50544836(CHEMBL4639640)
Affinity DataIC50: 3.5nMAssay Description:Displacement of [125I]MIP-1095 from PSMA in human PC3-PIP cells after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50544837(CHEMBL4648379)
Affinity DataIC50: 4.70nMAssay Description:Displacement of [125I]MIP-1095 from PSMA in human PC3-PIP cells after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50544833(Vipivotide tetraxetan | PSMA-617 | US20240366813, ...)
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]MIP-1095 from PSMA in human PC3-PIP cells after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetGlutamate carboxypeptidase 2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50544838(CHEMBL4635514)
Affinity DataIC50: 13nMAssay Description:Displacement of [125I]MIP-1095 from PSMA in human PC3-PIP cells after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed