Found 6 Enz. Inhib. hit(s) with all data for entry = 50011142 TargetProteinase-activated receptor 1(Homo sapiens (Human))
Hebei University Of Technology
Curated by ChEMBL
Hebei University Of Technology
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Hebei University Of Technology
Curated by ChEMBL
Hebei University Of Technology
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Hebei University Of Technology
Curated by ChEMBL
Hebei University Of Technology
Curated by ChEMBL
Affinity DataIC50: 550nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Hebei University Of Technology
Curated by ChEMBL
Hebei University Of Technology
Curated by ChEMBL
Affinity DataIC50: 610nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Hebei University Of Technology
Curated by ChEMBL
Hebei University Of Technology
Curated by ChEMBL
Affinity DataIC50: 760nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
TargetProteinase-activated receptor 1(Homo sapiens (Human))
Hebei University Of Technology
Curated by ChEMBL
Hebei University Of Technology
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human PAR1 expressed in KNRK cells assessed as inhibition of agonist-induced intracellular calcium mobilization by fluorimetri...More data for this Ligand-Target Pair
