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Found 58 Enz. Inhib. hit(s) with all data for entry = 50007996
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514737(CHEMBL4482861)
Affinity DataKi:  0.0417nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514738(CHEMBL4536304)
Affinity DataKi:  0.0537nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514722(CHEMBL4438801)
Affinity DataKi:  0.0661nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514727(CHEMBL4483022)
Affinity DataKi:  0.324nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514724(CHEMBL4535472)
Affinity DataKi:  0.977nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514745(CHEMBL4439953)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514739(CHEMBL4467833)
Affinity DataKi:  4.5nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514718(CHEMBL4438158)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514734(CHEMBL4568994)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514743(CHEMBL4454147)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514751(CHEMBL4554450)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50086502(2-BFi | 2-Benzofuran-2-yl-4,5-dihydro-1H-imidazole...)
Affinity DataKi:  229nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514721(CHEMBL4450506)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514721(CHEMBL4450506)
Affinity DataKi:  537nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514730(CHEMBL4456882)
Affinity DataKi:  603nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514731(CHEMBL4528557)
Affinity DataKi:  708nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514725(CHEMBL4459090)
Affinity DataKi:  1.18E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514742(CHEMBL4587519)
Affinity DataKi:  1.41E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514746(CHEMBL4587003)
Affinity DataKi:  2.24E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514728(CHEMBL4533687)
Affinity DataKi:  3.72E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514750(CHEMBL4475933)
Affinity DataKi:  4.57E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514747(CHEMBL151697)
Affinity DataKi:  6.76E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514729(CHEMBL4459403)
Affinity DataKi:  6.92E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514719(CHEMBL4590209)
Affinity DataKi:  7.59E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514726(CHEMBL4546903)
Affinity DataKi:  9.55E+3nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514741(CHEMBL4476557)
Affinity DataKi:  1.86E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514723(CHEMBL4534152)
Affinity DataKi:  2.57E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50226966(CHEMBL41103)
Affinity DataKi:  4.27E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  4.68E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514733(CHEMBL4445396)
Affinity DataKi:  4.90E+4nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514720(CHEMBL4469237)
Affinity DataKi:  1.15E+5nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514735(CHEMBL4584406)
Affinity DataKi:  1.41E+5nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514744(CHEMBL4434967)
Affinity DataKi:  1.70E+5nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514732(CHEMBL4553853)
Affinity DataKi:  3.63E+5nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514736(CHEMBL4465834)
Affinity DataKi:  4.17E+5nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514721(CHEMBL4450506)
Affinity DataKi:  9.12E+5nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514748(CHEMBL4527478)
Affinity DataKi: <1.00E+6nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514749(CHEMBL4543019)
Affinity DataKi: <1.00E+6nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514740(CHEMBL4531381)
Affinity DataKi: <1.00E+6nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM113058(US8633208, 1)
Affinity DataKi:  2.24E+6nMAssay Description:Displacement of [3H]RX821002 from alpha2-AR in human brain frontal cortex incubated for 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50050093((4-Chloro-6-methoxy-2-methyl-pyrimidin-5-yl)-imida...)
Affinity DataIC50:  3.5nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514738(CHEMBL4536304)
Affinity DataIC50:  8.10nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514744(CHEMBL4434967)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514724(CHEMBL4535472)
Affinity DataIC50:  29nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514719(CHEMBL4590209)
Affinity DataIC50:  65nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514737(CHEMBL4482861)
Affinity DataIC50:  182nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514725(CHEMBL4459090)
Affinity DataIC50:  646nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514718(CHEMBL4438158)
Affinity DataIC50:  1.35E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514726(CHEMBL4546903)
Affinity DataIC50:  3.39E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
University Of Barcelona

Curated by ChEMBL
LigandPNGBDBM50514722(CHEMBL4438801)
Affinity DataIC50:  5.50E+3nMAssay Description:Displacement of [3H]clonidine from I1IR in human brain frontal cortex in presence of adrenaline incubated for 45 mins by liquid scintillation spectro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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